SCHEMBL5525613

SCHEMBL5525613

CC(C)(C)c1nc(Cc2ccc(F)cc2Cl)c(C(=O)O)s1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 15/20 0.40
BCKDK O14874 1/20 0.38
TRPV1 Q8NER1 1/20 0.37
NPC1 O15118 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5528337 0.88 NPC1 (0.45) NPC1RAB9ASMN1; SMN2
SCHEMBL13494106 0.84 CYP1A2 (0.43) P2RX7BCKDKNPC1CYP1A2CYP2C19
SCHEMBL5520108 0.83 POLB (0.39) NPC1RAB9ASMN1; SMN2
SCHEMBL10266407 0.82 P2RX7 (0.39) P2RX7BCKDKNPC1CYP1A2CYP2C19
SCHEMBL5524260 0.80 PPARA (0.40) RAB9ASMN1; SMN2
SCHEMBL5521998 0.79 HCAR2 (0.46) TRPV1NPC1RAB9ASMN1; SMN2
SCHEMBL5524256 0.78 RAB9A (0.43) NPC1RAB9ASMN1; SMN2
SCHEMBL5520215 0.76 ALDH1A1 (0.41) NPC1SMN1; SMN2
SCHEMBL5522175 0.75 SMN1; SMN2 (0.41) NPC1RAB9ASMN1; SMN2
SCHEMBL5522358 0.75 RAB9A (0.51) NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120108565-A1 PYRROLE CARBOXYLIC ACID DERIVATIVES AS ANTIBACTERIAL AGENTS RANBAXY LABORATORIES LIMITED (IN) 2012-05-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120108565-A1 PYRROLE CARBOXYLIC ACID DERIVATIVES AS ANTIBACTERIAL AGENTS POLI, POLB, POLA1 P2RX7 2375/4885BCKDK 554/4885TRPV1 4123/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.