SCHEMBL5530335

SCHEMBL5530335

CCN1C[C@H](C)N(C=C(C(=O)O)C(=O)O)CC1=O

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
INMT O95050 1/20 0.30
CACNA1G O43497 2/20 0.30
CACNA1H O95180 2/20 0.30
CACNA1I Q9P0X4 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3985599 0.83 NPSR1 (0.34)
SCHEMBL3985687 0.74 CACNA1G (0.39) INMTCACNA1GCACNA1HCACNA1I
SCHEMBL8293964 0.60 POLB (0.67)
SCHEMBL9834992 0.60 F2 (0.38) INMT
SCHEMBL19546254 0.60 F2 (0.38) INMT
SCHEMBL867969 0.58
SCHEMBL13472137 0.58 POLB (0.46)
SCHEMBL17294311 0.58 BRD4 (0.42)
SCHEMBL14423078 0.58
SCHEMBL21011630 0.57 OPRM1 (0.35) INMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756114-B1 HIV INTEGRASE INHIBITORS MERCK SHARP & DOHME (US) 2014-11-19 EP disclosed
EP-1756114-A2 HIV INTEGRASE INHIBITORS Merck and Co., Inc. (US) 2007-02-28 EP disclosed
WO-2005110414-A2 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2005-11-24 WO disclosed