SCHEMBL5533509

SCHEMBL5533509

COC(=O)C[C@@H]1C[C@H](C/C=C(\C)CC#N)NC1=O

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.33
IRAK4 Q9NWZ3 2/20 0.31
ITGB3 P05106 1/20 0.31
ITGA2B P08514 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5533516 1.00 GAA (0.33) GAAIRAK4ITGB3ITGA2B
SCHEMBL5533521 1.00 GAA (0.33) GAAIRAK4ITGB3ITGA2B
SCHEMBL7275658 0.74 GAA (0.42) GAAIRAK4ITGB3ITGA2B
SCHEMBL7277780 0.73 GAA (0.41) GAAIRAK4ITGB3ITGA2B
SCHEMBL7282562 0.70 ITGB3 (0.56) IRAK4ITGB3ITGA2B
SCHEMBL7283083 0.70 ITGB3 (0.56) IRAK4ITGB3ITGA2B
SCHEMBL7276433 0.70 ITGB3 (0.56) IRAK4ITGB3ITGA2B
SCHEMBL7275480 0.68 GAA (0.37) GAAIRAK4ITGB3ITGA2B
SCHEMBL8863881 0.64 ITGB3 (0.43) IRAK4ITGB3ITGA2B
SCHEMBL3496534 0.64 KCNH2 (0.37) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1804793-A2 2-(ARYL)AZACYCLYLMETHYL CARBOXYLATES, SULFONATES, PHOSPHONATES, PHOSPHINATES AND HETEROCYCLES AS S1P RECEPTOR AGONISTS Merck & Co., Inc. (US) 2007-07-11 EP disclosed
WO-2006047195-A2 2-(ARYL)AZACYCLYLMETHYL CARBOXYLATES, SULFONATES, PHOSPHONATES, PHOSPHINATES AND HETEROCYCLES AS S1P RECEPTOR AGONISTS MERCK & CO., INC. (US) 2006-05-04 WO disclosed