SCHEMBL5533679

SCHEMBL5533679

Cc1c(CNC2CCN(C(=O)OC(C)(C)C)CC2)ccc2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.46
CCR8 P51685 1/20 0.46
KDM4E B2RXH2 2/20 0.46
PKM P14618 1/20 0.46
ALDH1A1 P00352 2/20 0.45
GPR119 Q8TDV5 3/20 0.45
NPC1 O15118 1/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
RAB9A P51151 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
STS P08842 1/20 0.44
EPHX2 P34913 1/20 0.43
KEAP1 Q14145 1/20 0.42
NFE2L2 Q16236 1/20 0.42
EPHX1 P07099 1/20 0.42
CHRM2 P08172 1/20 0.42
CHRM4 P08173 1/20 0.42
CHRM1 P11229 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5532244 0.89 ACHE (0.46) ACHECCR8KDM4EPKMALDH1A1
SCHEMBL20778605 0.81 GPR119 (0.50) KDM4EPKMALDH1A1GPR119NPC1
SCHEMBL2604335 0.79 KDM4E (0.53) CCR8KDM4EPKMALDH1A1GPR119
SCHEMBL69764 0.79 MAPT (0.54) KDM4EPKMALDH1A1GPR119NPC1
SCHEMBL31184445 0.79 KDM4E (0.53) CCR8KDM4EPKMALDH1A1GPR119
SCHEMBL69077 0.79 KDM4E (0.50) CCR8KDM4EPKMALDH1A1GPR119
SCHEMBL616004 0.79 STS (0.60) ACHEKDM4EPKMALDH1A1GPR119
SCHEMBL5992995 0.78 EPHX2 (0.56) KDM4EPKMALDH1A1GPR119NPC1
SCHEMBL4200062 0.78 MEN1 (0.57) ACHEKDM4EPKMALDH1A1GPR119
SCHEMBL16465018 0.78 EPHX2 (0.48) KDM4EPKMALDH1A1GPR119NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828122-A2 N-PYRROLIDIN-3-YL-AMIDE DERIVATIVES AS SEROTONIN AND NORADRENALIN RE-UPTAKE INHIBITORS Pfizer Limited (GB) 2007-09-05 EP disclosed
WO-2006064351-A2 N-PYRROLIDIN-3-YL-AMIDE DERIVATIVES AS SEROTONIN AND NORADRENALIN RE-UPTAKE INHIBITORS PFIZER LIMITED (GB) 2006-06-22 WO disclosed