SCHEMBL5532244

SCHEMBL5532244

CC(C)(C)OC(=O)N1CCC(NCc2ccc3ccccc3c2Br)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.46
KDM4E B2RXH2 1/20 0.45
PKM P14618 1/20 0.45
ALDH1A1 P00352 2/20 0.44
GPR119 Q8TDV5 2/20 0.44
BACE1 P56817 1/20 0.44
CCR8 P51685 1/20 0.44
NPC1 O15118 2/20 0.43
HTT P42858 2/20 0.43
RAB9A P51151 2/20 0.43
MAPT P10636 1/20 0.43
MAPK1 P28482 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
STS P08842 1/20 0.43
EPHX2 P34913 1/20 0.43
NCEH1 Q6PIU2 2/20 0.42
USP30 Q70CQ3 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5533679 0.89 ACHE (0.46) ACHEKDM4EPKMALDH1A1GPR119
SCHEMBL69077 0.83 KDM4E (0.50) KDM4EPKMALDH1A1GPR119CCR8
SCHEMBL69764 0.78 MAPT (0.54) KDM4EPKMALDH1A1GPR119NPC1
SCHEMBL31184445 0.78 KDM4E (0.53) KDM4EPKMALDH1A1GPR119CCR8
SCHEMBL2604335 0.78 KDM4E (0.53) KDM4EPKMALDH1A1GPR119CCR8
SCHEMBL616004 0.78 STS (0.60) ACHEKDM4EPKMALDH1A1GPR119
SCHEMBL4200062 0.78 MEN1 (0.57) ACHEKDM4EPKMALDH1A1GPR119
SCHEMBL5992995 0.78 EPHX2 (0.56) KDM4EPKMALDH1A1GPR119NPC1
SCHEMBL5013239 0.76 ALDH1A1 (0.51) KDM4EPKMALDH1A1GPR119NPC1
SCHEMBL20766458 0.75 GPR119 (0.52) KDM4EPKMALDH1A1GPR119NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828122-A2 N-PYRROLIDIN-3-YL-AMIDE DERIVATIVES AS SEROTONIN AND NORADRENALIN RE-UPTAKE INHIBITORS Pfizer Limited (GB) 2007-09-05 EP disclosed
WO-2006064351-A2 N-PYRROLIDIN-3-YL-AMIDE DERIVATIVES AS SEROTONIN AND NORADRENALIN RE-UPTAKE INHIBITORS PFIZER LIMITED (GB) 2006-06-22 WO disclosed