SCHEMBL5534100

SCHEMBL5534100

COC(=O)c1ccccc1C(C)(C)C#N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.49
LMNA P02545 2/20 0.49
ALDH1A1 P00352 3/20 0.47
HSD17B10 Q99714 2/20 0.47
CFTR P13569 1/20 0.47
KDM4E B2RXH2 4/20 0.47
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA5A P35218 1/20 0.46
CA9 Q16790 1/20 0.46
POLB P06746 1/20 0.46
ATM Q13315 1/20 0.46
KMT2A Q03164 2/20 0.42
MAPT P10636 1/20 0.42
ALOX15 P16050 1/20 0.42
SLC6A3 Q01959 4/20 0.41
MYC P01106 1/20 0.41
NR4A2 P43354 1/20 0.41
CREBBP Q92793 1/20 0.41
SLC6A4 P31645 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2193334 0.84 PDK2 (0.47) TSHRLMNAALDH1A1HSD17B10CFTR
SCHEMBL4987570 0.81 ALDH1A1 (0.46) TSHRLMNAALDH1A1HSD17B10KDM4E
SCHEMBL1788233 0.80 TSHR (0.57) TSHRLMNAALDH1A1HSD17B10CFTR
SCHEMBL4967948 0.79 ALDH1A1 (0.42) TSHRALDH1A1HSD17B10KDM4EATM
Ammonia Solution, Strong SCHEMBL28371090 0.79 TSHR (0.55) TSHRLMNAALDH1A1HSD17B10CFTR
SCHEMBL24895044 0.78 NR4A2 (0.47) TSHRALDH1A1HSD17B10CFTRKDM4E
SCHEMBL31676878 0.76 SLC6A3 (0.58) TSHRLMNAALDH1A1HSD17B10CFTR
SCHEMBL23354388 0.76 SLC6A3 (0.58) TSHRLMNAALDH1A1HSD17B10CFTR
SCHEMBL22745916 0.76 LMNA (0.52) TSHRLMNAALDH1A1HSD17B10CFTR
SCHEMBL10938198 0.75 TSHR (0.55) TSHRLMNAALDH1A1HSD17B10CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828147-A1 QUINOXALINES AS B-RAF INHIBITORS AstraZeneca AB (SE) 2007-09-05 EP disclosed
WO-2006040568-A1 QUINOXALINES AS B RAF INHIBITORS ASTRAZENECA AB (SE) 2006-04-20 WO disclosed