SCHEMBL5537419

SCHEMBL5537419

FC(F)(F)Oc1ccc(-c2[c]cccn2)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.47
GRIN2B Q13224 6/20 0.42
SUCNR1 Q9BXA5 1/20 0.41
MALT1 Q9UDY8 1/20 0.39
SLC1A5 Q15758 2/20 0.36
NOTUM Q6P988 1/20 0.36
CSF1R P07333 1/20 0.36
GRM2 Q14416 2/20 0.35
SCN3A Q9NY46 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5536136 0.86 FAAH (0.42) GRM2
SCHEMBL5536566 0.78 AHR (0.45) KMONOTUM
SCHEMBL5545405 0.77 KDM4E (0.45) GRIN2BNOTUM
SCHEMBL5542548 0.77 NISCH (0.42) KMOGRIN2B
SCHEMBL5545853 0.76 KMO (0.53) KMOGRIN2BSUCNR1MALT1SLC1A5
SCHEMBL14741867 0.72 KMO (0.51) KMOGRIN2BSLC1A5CSF1RGRM2
SCHEMBL29699525 0.71 KMO (0.51) KMOGRIN2BSLC1A5
SCHEMBL5535439 0.71 KMO (0.49) KMOGRIN2BSUCNR1SLC1A5NOTUM
SCHEMBL5537301 0.71 KMO (0.52) KMOGRIN2BSUCNR1SLC1A5NOTUM
SCHEMBL28158976 0.71 KMO (0.48) KMOGRIN2BSUCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2570418-A2 2,3-dihydro-6-nitroimidazo[2,1-b]oxazoles compound OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2013-03-20 EP disclosed
EP-1555267-B1 2,3-DIHYDRO-6-NITROIMIDAZO[2,1-b]OXAZOLES OTSUKA PHARMA CO LTD (JP) 2013-01-16 EP disclosed
US-7262212-B2 2,3-dihydro-6-nitroimidazo[2,1-b]oxazoles OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-08-28 US disclosed
US-20060094767-A1 2,3-Dihydro-6-nitroimidazo[2,1-b]oxazoles OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-05-04 US disclosed
EP-1555267-A1 2,3-DIHYDRO-6-NITROIMIDAZO 2,1-b OXAZOLES OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2005-07-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060094767-A1 2,3-Dihydro-6-nitroimidazo[2,1-b]oxazoles NR2C2, NR4A3, NR4A2 KMO 4404/4885GRIN2B 504/4885SUCNR1 152/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.