SCHEMBL5536136

SCHEMBL5536136

Fc1cc(-c2[c]cccn2)ccc1OC(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.42
PDE2A O00408 4/20 0.39
TRPM8 Q7Z2W7 3/20 0.39
SYK P43405 1/20 0.39
EPHX2 P34913 1/20 0.38
ALOX5AP P20292 1/20 0.38
FEN1 P39748 1/20 0.38
P2RX7 Q99572 3/20 0.36
SLC7A5 Q01650 1/20 0.35
CTSK P43235 1/20 0.34
NAAA Q02083 1/20 0.34
ABL1 P00519 1/20 0.34
GRM2 Q14416 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5537419 0.86 KMO (0.47) GRM2
SCHEMBL5541420 0.80 CYP17A1 (0.41)
SCHEMBL5545405 0.79 KDM4E (0.45)
SCHEMBL5547891 0.74 FAAH (0.44) FAAHPDE2ATRPM8SYKEPHX2
SCHEMBL28019370 0.73 GRIN1 (0.31)
SCHEMBL5542548 0.73 NISCH (0.42)
SCHEMBL5538786 0.73 ACHE (0.44) SYK
SCHEMBL28413182 0.73 GRIN2B (0.40)
SCHEMBL28138779 0.72 GRIN2B (0.39)
SCHEMBL1973038 0.71 MAPK14 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2570418-A2 2,3-dihydro-6-nitroimidazo[2,1-b]oxazoles compound OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2013-03-20 EP disclosed
EP-1555267-B1 2,3-DIHYDRO-6-NITROIMIDAZO[2,1-b]OXAZOLES OTSUKA PHARMA CO LTD (JP) 2013-01-16 EP disclosed
US-7262212-B2 2,3-dihydro-6-nitroimidazo[2,1-b]oxazoles OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-08-28 US disclosed
US-20060094767-A1 2,3-Dihydro-6-nitroimidazo[2,1-b]oxazoles OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-05-04 US disclosed
EP-1555267-A1 2,3-DIHYDRO-6-NITROIMIDAZO 2,1-b OXAZOLES OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2005-07-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060094767-A1 2,3-Dihydro-6-nitroimidazo[2,1-b]oxazoles NR2C2, NR4A3, NR4A2 FAAH 4363/4885PDE2A 4223/4885TRPM8 3538/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.