SCHEMBL5540930

SCHEMBL5540930

CC(C)C(C)(C)C(=O)NCCc1ccc(OCc2ccccc2)c(OCc2ccccc2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.54
MTNR1B P49286 2/20 0.54
SLC2A1 P11166 1/20 0.50
ALDH1A1 P00352 3/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
ABCB1 P08183 1/20 0.48
ABCG2 Q9UNQ0 1/20 0.48
OPRK1 P41145 2/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
LMNA P02545 1/20 0.48
POLB P06746 1/20 0.48
HTT P42858 1/20 0.48
OPRD1 P41143 1/20 0.47
BCHE P06276 2/20 0.47
FFAR4 Q5NUL3 1/20 0.46
APP P05067 1/20 0.46
NPC1 O15118 1/20 0.45
PKM P14618 1/20 0.45
RAB9A P51151 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2746596 0.86 MTNR1A (0.56) MTNR1AMTNR1BSLC2A1ALDH1A1MEN1
SCHEMBL25300742 0.84 MTNR1A (0.56) MTNR1AMTNR1BSLC2A1ALDH1A1MEN1
SCHEMBL30517507 0.84 MTNR1A (0.56) MTNR1AMTNR1BSLC2A1ALDH1A1MEN1
SCHEMBL7281747 0.83 MTNR1A (0.55) MTNR1AMTNR1BSLC2A1ALDH1A1MEN1
SCHEMBL13774782 0.81 OPRK1 (0.68) ALDH1A1MEN1KMT2AOPRK1SMN1; SMN2
SCHEMBL5543465 0.81 CA12 (0.61) ALDH1A1MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL10163435 0.80 MTNR1A (0.62) MTNR1AMTNR1BSLC2A1ALDH1A1MEN1
SCHEMBL12707505 0.80 SLC2A1 (0.58) MTNR1AMTNR1BSLC2A1ALDH1A1MEN1
SCHEMBL441815 0.80 MTNR1A (0.65) MTNR1AMTNR1BALDH1A1MEN1KMT2A
SCHEMBL441779 0.80 MTNR1A (0.59) MTNR1AMTNR1BALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed