SCHEMBL5541772

SCHEMBL5541772

CC(C)(C)CNC(=O)Nc1ccc(C(=O)O)cc1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 5/20 0.61
NR1H4 Q96RI1 1/20 0.61
NAMPT P43490 2/20 0.54
CA12 O43570 1/20 0.48
CA2 P00918 1/20 0.48
CA9 Q16790 1/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
FAAH O00519 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
NPC1 O15118 1/20 0.45
MAPT P10636 1/20 0.45
RAB9A P51151 1/20 0.45
TAAR1 Q96RJ0 1/20 0.45
ALDH1A1 P00352 1/20 0.45
CNR1 P21554 1/20 0.44
MITF O75030 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12127864 0.84 SMN1; SMN2 (0.59) EPHX2MEN1KMT2ASMN1; SMN2NPC1
SCHEMBL23453358 0.83 NPC1 (0.62) MEN1KMT2ACYP1A2CYP2C9SMN1; SMN2
SCHEMBL14679305 0.81 CASR (0.59) CA12CA2CA9MEN1KMT2A
SCHEMBL20589556 0.81 FPR2 (0.47) EPHX2NAMPTCA12CA2CA9
SCHEMBL19818490 0.81 RAB9A (0.60) EPHX2NR1H4CA12CA2CA9
SCHEMBL13614142 0.81 NAMPT (0.58) EPHX2NR1H4NAMPTCA12CA2
SCHEMBL19964254 0.79 EPHX2 (0.50) EPHX2NR1H4CA2MEN1KMT2A
SCHEMBL18026623 0.79 HDAC3 (0.56) NAMPTCA12CA2CA9MEN1
SCHEMBL3762312 0.78 MEN1 (0.62) EPHX2NR1H4NAMPTMEN1KMT2A
SCHEMBL4745756 0.78 EPHX2 (0.71) EPHX2NR1H4CA12CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed