SCHEMBL5542596

SCHEMBL5542596

CCN(CC)C(=O)CNC(=O)C(C)(C)C(C)C

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.36
CA12 O43570 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA9 Q16790 2/20 0.33
PRMT3 O60678 1/20 0.32
HSD17B10 Q99714 1/20 0.31
DPP4 P27487 1/20 0.30
MMP8 P22894 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11922838 0.81 LMNA (0.41) LMNACA12CA1CA2CA9
SCHEMBL5541518 0.75 ALDH1A1 (0.47) LMNA
SCHEMBL18907822 0.74 MMP8 (0.34) MMP8
SCHEMBL10266048 0.73 TET2 (0.47) LMNACA12CA1CA2CA9
SCHEMBL19981641 0.73 ALDH1A1 (0.46) LMNACA12CA1CA2CA9
SCHEMBL5541412 0.72 PIK3CD (0.33) LMNA
SCHEMBL24869141 0.70 LMNA (0.46) LMNACA12CA1CA2CA9
SCHEMBL18909748 0.69 CYP2D6 (0.50) HSD17B10MMP8
SCHEMBL13712976 0.69 LMNA (0.44) LMNACA12CA1CA2CA9
SCHEMBL23197920 0.68 EPHX1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed