SCHEMBL5543524

SCHEMBL5543524

CC(C)(C)c1cn2c(=O)[nH]nc2c(NCCc2ccc(O)cc2)n1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.43
GSK3B P49841 12/20 0.43
GSK3A P49840 11/20 0.41
TTBK1 Q5TCY1 1/20 0.36
TTBK2 Q6IQ55 1/20 0.36
GPR84 Q9NQS5 1/20 0.36
ILK Q13418 1/20 0.36
ESRRB O95718 2/20 0.36
ESRRG P62508 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5543493 0.89 GSK3B (0.50) ADORA1GSK3BGSK3AGPR84
SCHEMBL3528033 0.88 GSK3B (0.56) ADORA1GSK3BGSK3A
SCHEMBL5545429 0.88 GSK3B (0.46) ADORA1GSK3BGSK3A
SCHEMBL5549014 0.87 CA1 (0.49) ADORA1
SCHEMBL5545525 0.85 ADORA1 (0.47) ADORA1GSK3BGSK3A
SCHEMBL3526786 0.85 GSK3B (0.56) ADORA1GSK3BGSK3A
SCHEMBL5549261 0.84 KMT2A (0.48)
SCHEMBL3529268 0.83 ADORA1 (0.37) ADORA1GSK3BGSK3A
SCHEMBL5545556 0.83 GSK3A (0.48) ADORA1GSK3BGSK3A
SCHEMBL3525610 0.82 GSK3B (0.55) ADORA1GSK3BGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed