SCHEMBL5543567

SCHEMBL5543567

CC(C)(C)c1cn2c(=O)[nH]nc2c(NCCCCc2ccccc2)n1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.47
GSK3A P49840 14/20 0.45
GSK3B P49841 14/20 0.45
TYMP P19971 1/20 0.41
GPR84 Q9NQS5 1/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5545556 0.97 GSK3A (0.48) ADORA1GSK3AGSK3B
SCHEMBL5545525 0.84 ADORA1 (0.47) ADORA1GSK3AGSK3B
SCHEMBL3528033 0.83 GSK3B (0.56) ADORA1GSK3AGSK3B
SCHEMBL5545476 0.82 ADORA1 (0.39) ADORA1GSK3AGSK3B
SCHEMBL5543524 0.82 ADORA1 (0.43) ADORA1GSK3AGSK3BGPR84
SCHEMBL5543505 0.82 GSK3A (0.36) GSK3AGSK3B
SCHEMBL3525610 0.82 GSK3B (0.55) ADORA1GSK3AGSK3B
SCHEMBL5549283 0.81 GSK3B (0.58) ADORA1GSK3AGSK3B
SCHEMBL3527204 0.81 GSK3A (0.41) GSK3AGSK3B
SCHEMBL5545429 0.80 GSK3B (0.46) ADORA1GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed