SCHEMBL5543693

SCHEMBL5543693

CC(C)C(C)(C)C(=O)NS(=O)(=O)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 3/20 0.52
MITF O75030 2/20 0.50
HPGD P15428 2/20 0.50
LARS1 Q9P2J5 1/20 0.50
LMNA P02545 1/20 0.50
KMT2A Q03164 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.47
GPR55 Q9Y2T6 1/20 0.47
CA2 P00918 2/20 0.46
KDM4E B2RXH2 2/20 0.45
PTGS1 P23219 1/20 0.45
PTGS2 P35354 1/20 0.45
BCAT1 P54687 1/20 0.45
MMP2 P08253 2/20 0.44
CA1 P00915 1/20 0.44
MMP1 P03956 1/20 0.44
MMP9 P14780 1/20 0.44
MMP8 P22894 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14212012 0.85 NLRP3 (0.49) LMNAKMT2ASMN1; SMN2CA2PTGS1
SCHEMBL5537015 0.84 HTT (0.59) KMT2ASMN1; SMN2MAPTHTTBCAT1
SCHEMBL13764330 0.82 PPARA (0.57) PPARAMITFHPGDLARS1LMNA
SCHEMBL29317683 0.80 PPARA (0.59) PPARAMITFHPGDLARS1LMNA
SCHEMBL3531889 0.79 PPARA (0.55) PPARAMITFHPGDLARS1LMNA
SCHEMBL4584839 0.79 PPARA (0.55) PPARAMITFHPGDLARS1LMNA
SCHEMBL85199 0.75 ALDH1A1 (0.69) MITFHPGDLARS1LMNAKMT2A
SCHEMBL5394506 0.75 CA1 (0.57) PPARAHPGDLARS1CA2KDM4E
SCHEMBL14278270 0.74 PPARA (0.56) PPARALARS1KMT2ASMN1; SMN2CA2
SCHEMBL27907157 0.73 ALDH1A1 (0.48) PPARAMITFHPGDLARS1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed