SCHEMBL5545017

SCHEMBL5545017

O=C(NC1=NCC2=CN(C(=O)c3sc4ccccc4c3Cl)CCC2=N1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
LMNA P02545 2/20 0.41
KMT2A Q03164 2/20 0.41
NPC1 O15118 2/20 0.41
MAPT P10636 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
PRSS12 P56730 12/20 0.40
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
MCL1 Q07820 1/20 0.38
OGG1 O15527 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5545011 0.73 NPC1 (0.41) ALDH1A1LMNAKMT2ANPC1MAPT
SCHEMBL5538119 0.66 RAB9A (0.46) ALDH1A1LMNAKMT2ANPC1MAPT
SCHEMBL5546870 0.66 NAMPT (0.34) ALDH1A1LMNAKMT2ANPC1MAPT
SCHEMBL5548741 0.65 SMN1; SMN2 (0.41) ALDH1A1LMNAKMT2ANPC1MAPT
SCHEMBL3533825 0.65 PDGFRB (0.50) ALDH1A1LMNAKMT2AMAPTKDM4E
SCHEMBL5546603 0.63 HPGDS (0.39) ALDH1A1LMNAKMT2ANPC1MAPT
SCHEMBL5548490 0.63 MAPT (0.39) ALDH1A1KMT2AMAPTRAB9ASMN1; SMN2
SCHEMBL14246804 0.62 ALDH1A1 (0.68) ALDH1A1LMNAKMT2ANPC1MAPT
SCHEMBL11177633 0.61 MCL1 (0.72) ALDH1A1LMNAKMT2ANPC1MAPT
SCHEMBL14246928 0.61 ALDH1A1 (0.67) ALDH1A1LMNAKMT2ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed