SCHEMBL5545113

SCHEMBL5545113

Oc1nccc2sc(-c3ncco3)cc12

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.33
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
HPGDS O60760 1/20 0.31
BRD4 O60885 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5537255 0.72 KDM4E (0.50)
SCHEMBL7916406 0.71 IKBKB (0.46) LTA4HADORA2AADORA1HPGDS
SCHEMBL5342853 0.69 ALDH1A1 (0.39)
SCHEMBL30633034 0.68 MEN1 (0.39) LTA4HADORA2AADORA1HPGDS
SCHEMBL30632958 0.68 ADRA1A (0.36) LTA4HADORA2AADORA1HPGDS
SCHEMBL3040416 0.67 NPC1 (0.46) ADORA2AADORA1
SCHEMBL31128921 0.67 APP (0.47)
SCHEMBL7058872 0.65 PIM1 (0.66)
SCHEMBL29700510 0.63 ALDH1A1 (0.34) ADORA2AADORA1BRD4
SCHEMBL5030066 0.62 LTA4H (0.39) LTA4HADORA2AADORA1HPGDSBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1805187-A1 INHIBITORS OF HEPATITIS C VIRUS PROTEASE, AND COMPOSITIONS AND TREATMENTS USING THE SAME Pfizer, Inc. (US) 2007-07-11 EP disclosed
WO-2006043145-A1 INHIBITORS OF HEPATITIS C VIRUS PROTEASE, AND COMPOSITIONS AND TREATMENTS USING THE SAME PFIZER INC. (US) 2006-04-27 WO disclosed