SCHEMBL5545549

SCHEMBL5545549

CC(C)(C)c1cn2c(=O)[nH]nc2c(NCCc2cccs2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.43
CASP3 P42574 1/20 0.43
CASP7 P55210 1/20 0.43
CASP8 Q14790 1/20 0.43
GPR84 Q9NQS5 1/20 0.42
PTGS2 P35354 1/20 0.38
ADORA1 P30542 2/20 0.38
GSK3B P49841 7/20 0.37
PDE4B Q07343 2/20 0.37
CHRM3 P20309 1/20 0.37
PDE4A P27815 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
GSK3A P49840 6/20 0.36
HRH4 Q9H3N8 1/20 0.36
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
RECQL P46063 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5543068 0.90 SMN1; SMN2 (0.41) PTGS2ADORA1MEN1LMNAPOLB
SCHEMBL5543318 0.82 MEN1 (0.40) ADORA1GSK3BGSK3AMEN1KMT2A
SCHEMBL3528033 0.82 GSK3B (0.56) ADORA1GSK3BGSK3A
SCHEMBL5545517 0.80 GSK3B (0.54) ADORA1GSK3BGSK3ALMNARAB9A
SCHEMBL5549402 0.79 ADORA1 (0.43) GPR84ADORA1GSK3BGSK3AMEN1
SCHEMBL5543493 0.79 GSK3B (0.50) GPR84ADORA1GSK3BGSK3AMAPT
SCHEMBL5543524 0.79 ADORA1 (0.43) GPR84ADORA1GSK3BGSK3A
SCHEMBL5545556 0.79 GSK3A (0.48) ADORA1GSK3BGSK3A
SCHEMBL3521775 0.79 GSK3B (0.36) ADORA1GSK3BGSK3A
SCHEMBL5545590 0.79 GSK3B (0.35) ADORA1GSK3BGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed