SCHEMBL5546357

SCHEMBL5546357

CCC([n+]1c2ccccc2cc2ccccc21)S(=O)(=O)O

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ATM Q13315 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
RAB9A P51151 1/20 0.41
NPC1 O15118 1/20 0.39
CYP2D6 P10635 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
TERT O14746 1/20 0.31
ALDH1A1 P00352 2/20 0.31
TSHR P16473 1/20 0.31
GAA P10253 2/20 0.30
KDM4E B2RXH2 1/20 0.30
HPGD P15428 1/20 0.30
NR1I2 O75469 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9011152 0.83 KDM4E (0.42) MEN1KMT2ACYP2D6HSD17B10TAS1R3
SCHEMBL8497616 0.80 KDM4E (0.33) MEN1KMT2AALDH1A1GAAKDM4E
SCHEMBL9011089 0.76 MEN1 (0.42) MEN1KMT2ARAB9ANPC1ALDH1A1
SCHEMBL5134000 0.75
SCHEMBL16859490 0.70 ATM (0.47) ATMMEN1KMT2ARAB9ANPC1
Anthracene SCHEMBL27663468 0.70 HTR2A (0.42) MEN1KMT2ARAB9ACYP2D6HSD17B10
SCHEMBL9010948 0.68 MEN1 (0.40) ATMMEN1KMT2ARAB9ANPC1
SCHEMBL9010950 0.66 NPC1 (0.33) KMT2ARAB9ANPC1CYP2D6HSD17B10
SCHEMBL17157330 0.66 SLC22A2 (0.38) MEN1KMT2AALDH1A1KDM4EHPGD
SCHEMBL164734 0.64 ATM (0.46) ATMMEN1KMT2ARAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1088229-A4 HIGH THROUGHPUT METHODS, SYSTEMS AND APPARATUS FOR PERFORMING CELL BASED SCREENING ASSAYS CALIPER TECHN CORP (US) 2002-05-08 EP claimed
EP-1088229-A1 HIGH THROUGHPUT METHODS, SYSTEMS AND APPARATUS FOR PERFORMING CELL BASED SCREENING ASSAYS Caliper Technologies Corporation (US) 2001-04-04 EP claimed
WO-2000014515-A9 LOW FREQUENCY MODULATION SENSORS USING NANOSECOND FLUOROPHORES UNIV MARYLAND (US) 2000-08-31 WO claimed
WO-2000014515-A1 LOW FREQUENCY MODULATION SENSORS USING NANOSECOND FLUOROPHORES UNIVERSITY OF MARYLAND AT BALTIMORE (US) 2000-03-16 WO claimed
WO-1999067639-A1 HIGH THROUGHPUT METHODS, SYSTEMS AND APPARATUS FOR PERFORMING CELL BASED SCREENING ASSAYS CALIPER TECHNOLOGIES CORPORATION (US) 1999-12-29 WO claimed
WO-2024102758-A2 N-(N-AMINOALKYL)PHENANTHRIDIUNIUM SERIES OF CHLORIDE-SENSITIVE FLUOROPHORES AND METHODS OF USE THEREOF THE GENERAL HOSPITAL CORPORATION (US) 2024-05-16 WO disclosed
CN-112368265-A N-alkylation of 9, 10-dihydroacridines 美国西门子医学诊断股份有限公司 2021-02-12 CN disclosed
EP-1179087-B1 FOCUSING OF MICROPARTICLES IN MICROFLUIDIC SYSTEMS CALIPER LIFE SCIENCES INC (US) 2019-03-27 EP disclosed
EP-3173487-B1 DEVICE FOR DETECTION OF HALOGENATED HYDROCARBONS UNIV MASARYKOVA (CZ) 2019-02-20 EP disclosed
EP-3173487-A1 DEVICE FOR DETECTION OF HALOGENATED HYDROCARBONS Masarykova univerzita (CZ) 2017-05-31 EP disclosed
US-7276330-B2 Devices, systems and methods for time domain multiplexing of reagents CALIPER TECHNOLOGIES CORP. (US) 2007-10-02 US disclosed
EP-1147417-A4 DEVICES, SYSTEMS AND METHODS FOR TIME DOMAIN MULTIPLEXING OF REAGENTS CALIPER LIFE SCIENCES INC (US) 2006-06-28 EP disclosed
EP-1147417-A1 DEVICES, SYSTEMS AND METHODS FOR TIME DOMAIN MULTIPLEXING OF REAGENTS Caliper Technologies Corporation (US) 2001-10-24 EP disclosed
WO-2000045172-A9 DEVICES, SYSTEMS AND METHODS FOR TIME DOMAIN MULTIPLEXING OF REAGENTS CALIPER TECHN CORP (US) 2001-10-11 WO disclosed
EP-1088229-A1 HIGH THROUGHPUT METHODS, SYSTEMS AND APPARATUS FOR PERFORMING CELL BASED SCREENING ASSAYS Caliper Technologies Corporation (US) 2001-04-04 EP disclosed
WO-2000070080-A1 FOCUSING OF MICROPARTICLES IN MICROFLUIDIC SYSTEMS CALIPER TECHNOLOGIES CORP. (US) 2000-11-23 WO disclosed
WO-2000014515-A9 LOW FREQUENCY MODULATION SENSORS USING NANOSECOND FLUOROPHORES UNIV MARYLAND (US) 2000-08-31 WO disclosed
WO-2000045172-A1 DEVICES, SYSTEMS AND METHODS FOR TIME DOMAIN MULTIPLEXING OF REAGENTS CALIPER TECHNOLOGIES CORP. (US) 2000-08-03 WO disclosed
WO-2000014515-A1 LOW FREQUENCY MODULATION SENSORS USING NANOSECOND FLUOROPHORES UNIVERSITY OF MARYLAND AT BALTIMORE (US) 2000-03-16 WO disclosed
WO-1999067639-A1 HIGH THROUGHPUT METHODS, SYSTEMS AND APPARATUS FOR PERFORMING CELL BASED SCREENING ASSAYS CALIPER TECHNOLOGIES CORPORATION (US) 1999-12-29 WO disclosed