SCHEMBL5546559

SCHEMBL5546559

Cc1ccc(C(=O)N2C=C3CN=C(NC(=O)c4ccc(C(C)(C)C)cc4)N=C3CC2)cc1[N+](=O)[O-]

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.50
RAB9A P51151 5/20 0.50
LMNA P02545 4/20 0.50
MAPT P10636 3/20 0.50
MAPK1 P28482 3/20 0.50
ATM Q13315 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
HPGD P15428 3/20 0.41
HTT P42858 2/20 0.41
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
POLB P06746 3/20 0.40
GAA P10253 3/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
ALDH1A1 P00352 3/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
GLA P06280 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5543018 0.76 ALDH1A1 (0.43) NPC1RAB9ALMNAMAPTMAPK1
SCHEMBL5546556 0.75 LMNA (0.45) NPC1RAB9ALMNAMAPTMAPK1
SCHEMBL5546926 0.73 TDP1 (0.38) NPC1RAB9ALMNAMAPTATM
SCHEMBL5540355 0.68 CA1 (0.39) NPC1RAB9ALMNAMAPTATM
SCHEMBL3532849 0.68 LMNA (0.51) NPC1RAB9ALMNAMAPTMAPK1
SCHEMBL5537982 0.68 NPC1 (0.42) NPC1RAB9ALMNAMAPTHPGD
SCHEMBL5538068 0.67 MAPT (0.39) NPC1RAB9AMAPTKMT2A
SCHEMBL5546575 0.66 ADORA2A (0.36) MAPTMEN1KMT2APOLB
SCHEMBL5540370 0.62 MAPT (0.41) NPC1RAB9ALMNAMAPTMAPK1
SCHEMBL10126443 0.61 GAA (0.76) LMNAHPGDHTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed