SCHEMBL5543018

SCHEMBL5543018

CC(C)(C)c1ccc(C(=O)NC2=NCC3=CN(S(=O)(=O)c4ccc([N+](=O)[O-])cc4)CCC3=N2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
MAPT P10636 4/20 0.43
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HSD11B1 P28845 3/20 0.43
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
TRPV4 Q9HBA0 1/20 0.40
ATM Q13315 1/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
TUBA1B P68363 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5540355 0.81 CA1 (0.39) ALDH1A1MAPTNPC1RAB9ALMNA
SCHEMBL5545044 0.76 ALDH1A1 (0.44) ALDH1A1MAPTRAB9ALMNASMN1; SMN2
SCHEMBL5546559 0.76 NPC1 (0.50) ALDH1A1MAPTNPC1RAB9ALMNA
SCHEMBL5540370 0.71 MAPT (0.41) ALDH1A1MAPTNPC1RAB9ALMNA
SCHEMBL5540254 0.69 RAB9A (0.37) ALDH1A1MAPTRAB9ALMNASMN1; SMN2
SCHEMBL3528675 0.67 MAPT (0.47) ALDH1A1MAPTNPC1RAB9ALMNA
SCHEMBL7296723 0.66 RAB9A (0.71) ALDH1A1MAPTNPC1RAB9ALMNA
SCHEMBL1687869 0.66 RAB9A (0.71) ALDH1A1MAPTNPC1RAB9ALMNA
SCHEMBL7300836 0.66 RAB9A (0.71) ALDH1A1MAPTNPC1RAB9ALMNA
SCHEMBL5546926 0.66 TDP1 (0.38) ALDH1A1MAPTNPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed