SCHEMBL5547414

SCHEMBL5547414

O=C(O)C1CN(C(c2ccccc2)c2ccccc2)CCN1C(=O)CN(c1ccccc1)c1ccccc1

nearest known ligand 0.70

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 12/20 0.69
CACNB1 Q02641 12/20 0.69
CACNA1C Q13936 4/20 0.69
CACNA1A O00555 2/20 0.69
CACNA1B Q00975 10/20 0.64
SLC6A9 P48067 1/20 0.45
AGTR2 P50052 3/20 0.44
CACNA1H O95180 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4187829 0.83 CACNA2D1 (0.97) CACNA2D1CACNB1CACNA1CCACNA1ACACNA1B
SCHEMBL8239769 0.83 CACNA2D1 (0.75) CACNA2D1CACNB1CACNA1CCACNA1ACACNA1B
SCHEMBL5541405 0.78 CACNA2D1 (1.00) CACNA2D1CACNB1CACNA1CCACNA1BCACNA1H
SCHEMBL5269185 0.77 CACNA2D1 (0.66) CACNA2D1CACNB1CACNA1CCACNA1ACACNA1B
SCHEMBL7376496 0.76 ALDH1A1 (0.52) CACNA2D1CACNB1CACNA1B
SCHEMBL7376500 0.76 ALDH1A1 (0.52) CACNA2D1CACNB1CACNA1B
SCHEMBL5547670 0.74 CACNA2D1 (0.67) CACNA2D1CACNB1CACNA1CCACNA1ACACNA1B
SCHEMBL5268550 0.73 CACNA2D1 (0.80) CACNA2D1CACNB1CACNA1CCACNA1ACACNA1B
SCHEMBL5544042 0.72 CACNA2D1 (1.00) CACNA2D1CACNB1CACNA1CCACNA1ACACNA1B
SCHEMBL6507611 0.72 CACNA2D1 (0.85) CACNA2D1CACNB1CACNA1CCACNA1ACACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745042-A1 DIARYLAMINE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS Neuromed Pharmaceuticals, Ltd. (CA) 2007-01-24 EP claimed
WO-2005097779-A1 DIARYLAMINE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS NEUROMED PHARMACEUTICALS LTD. (CA) 2005-10-20 WO claimed