SCHEMBL5547439

SCHEMBL5547439

COc1ccc(C(c2ccc(C(F)(F)F)cc2)N2CCN(C(C=O)N(c3ccccc3)c3ccccc3)CC2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 4/20 0.58
CACNB1 Q02641 4/20 0.58
CACNA1A O00555 2/20 0.58
CACNA1B Q00975 3/20 0.45
CACNA1C Q13936 3/20 0.45
CACNA1G O43497 2/20 0.45
CCR3 P51677 2/20 0.45
OPRD1 P41143 4/20 0.45
OPRM1 P35372 3/20 0.45
OPRK1 P41145 3/20 0.45
OPRL1 P41146 3/20 0.45
CYP2D6 P10635 3/20 0.44
CYP3A4 P08684 2/20 0.40
CYP3A5 P20815 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HTR1A P08908 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
USP2 O75604 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5547413 0.78 CACNA2D1 (0.74) CACNA2D1CACNB1CACNA1ACACNA1BCACNA1C
SCHEMBL5547408 0.78 CACNA2D1 (0.65) CACNA2D1CACNB1CACNA1ACACNA1BCACNA1C
SCHEMBL4189200 0.77 CACNA2D1 (0.59) CACNA2D1CACNB1CACNA1ACACNA1BCACNA1C
SCHEMBL5547650 0.74 CHRM2 (0.57) CACNA2D1CACNB1CACNA1ACACNA1BCACNA1C
SCHEMBL4179716 0.74 CACNA2D1 (1.00) CACNA2D1CACNB1CACNA1ACACNA1BCACNA1C
SCHEMBL3426145 0.73 CACNA2D1 (0.70) CACNA2D1CACNB1CACNA1ACACNA1BCACNA1C
SCHEMBL8305212 0.71 CACNA2D1 (0.54) CACNA2D1CACNB1CACNA1ACACNA1BCACNA1C
SCHEMBL7493410 0.69 CYP1A1 (0.48) CACNA2D1CACNB1CACNA1AOPRK1MEN1
SCHEMBL5549077 0.69 CACNA2D1 (0.58) CACNA2D1CACNB1CACNA1BCACNA1CCACNA1G
SCHEMBL5541529 0.68 CACNA2D1 (0.58) CACNA2D1CACNB1CACNA1BCACNA1CCACNA1G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745042-A1 DIARYLAMINE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS Neuromed Pharmaceuticals, Ltd. (CA) 2007-01-24 EP claimed
WO-2005097779-A1 DIARYLAMINE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS NEUROMED PHARMACEUTICALS LTD. (CA) 2005-10-20 WO claimed