SCHEMBL5548494

SCHEMBL5548494

O=c1[nH]nc2c(NCCc3c[nH]c4ccccc34)nc(-c3ccccc3)cn12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.47
POLB P06746 1/20 0.47
SLC2A1 P11166 1/20 0.47
RAD52 P43351 1/20 0.47
GPR18 Q14330 7/20 0.47
GBA1 P04062 1/20 0.47
GPR84 Q9NQS5 1/20 0.47
LMNA P02545 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
MEN1 O00255 2/20 0.45
ALDH1A1 P00352 1/20 0.45
HTR6 P50406 2/20 0.45
ILK Q13418 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
PAK4 O96013 1/20 0.43
MAPT P10636 1/20 0.43
MAPK1 P28482 1/20 0.43
HTT P42858 1/20 0.43
GFER P55789 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5545434 0.84 GPR18 (0.46) KMT2APOLBSLC2A1RAD52GPR18
SCHEMBL5355790 0.72 ADORA1 (0.53) KMT2APOLBSLC2A1RAD52GPR18
SCHEMBL5354834 0.72 ADORA1 (0.53) KMT2APOLBSLC2A1RAD52GPR18
SCHEMBL5545544 0.72 TRPM8 (0.49) KMT2APOLBMEN1MAPT
SCHEMBL21248401 0.70 GBA1 (0.45) KMT2APOLBSLC2A1RAD52GPR18
SCHEMBL3524781 0.70 CLK4 (0.45) KMT2ALMNASMN1; SMN2MEN1ALDH1A1
SCHEMBL21248476 0.70 GBA1 (0.44) KMT2APOLBSLC2A1RAD52GPR18
SCHEMBL5549374 0.70 METAP1 (0.42) NPC1RAB9ADRD2
SCHEMBL21092866 0.69 GBA1 (0.44) KMT2APOLBSLC2A1RAD52GPR18
SCHEMBL21093186 0.69 GBA1 (0.43) KMT2APOLBSLC2A1RAD52GPR18

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed