SCHEMBL5548616

SCHEMBL5548616

COc1cccc(CCNc2nc(C(C)(C)C)cn3c(=O)[nH]nc23)c1OC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA14 Q9ULX7 1/20 0.40
GSK3B P49841 6/20 0.39
GSK3A P49840 5/20 0.39
PARP1 P09874 1/20 0.36
ADORA1 P30542 1/20 0.36
GAA P10253 3/20 0.35
KDM4E B2RXH2 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
TSHR P16473 1/20 0.34
CRHBP P24387 1/20 0.34
MAPK1 P28482 1/20 0.34
CRHR2 Q13324 1/20 0.34
LMNA P02545 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HTR2A P28223 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5549283 0.81 GSK3B (0.58) GSK3BGSK3AADORA1KDM4E
SCHEMBL3529299 0.81 GSK3B (0.41) GSK3BGSK3AADORA1
SCHEMBL5549261 0.81 KMT2A (0.48) GAAKDM4ESMN1; SMN2POLBTSHR
SCHEMBL5545429 0.81 GSK3B (0.46) GSK3BGSK3AADORA1LMNA
SCHEMBL5543514 0.79 GSK3B (0.40) GSK3BGSK3AADORA1KDM4ESMN1; SMN2
SCHEMBL5549416 0.78 PDE5A (0.40) GSK3BGSK3AGAAKDM4ESMN1; SMN2
SCHEMBL3527695 0.77 GSK3B (0.42) GSK3BGSK3AADORA1POLBTSHR
SCHEMBL5545434 0.77 GPR18 (0.46) KDM4ESMN1; SMN2ALDH1A1POLBMAPK1
SCHEMBL5543318 0.77 MEN1 (0.40) GSK3BGSK3AADORA1
SCHEMBL3528033 0.77 GSK3B (0.56) GSK3BGSK3AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed