SCHEMBL5550132

SCHEMBL5550132

CC(=O)NCCNc1nc(C(C)(C)C)cn2c(=O)[nH]nc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ILK Q13418 2/20 0.35
CA12 O43570 1/20 0.34
CA4 P22748 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
GLP1R P43220 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ADORA1 P30542 2/20 0.33
ADORA2A P29274 1/20 0.33
IKBKB O14920 1/20 0.33
CHUK O15111 1/20 0.33
GSK3B P49841 7/20 0.33
GSK3A P49840 6/20 0.33
CYP1A2 P05177 4/20 0.33
CYP2D6 P10635 4/20 0.33
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 1/20 0.33
ALOX15 P16050 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3529957 0.87 BRD4 (0.45) ALDH1A1
SCHEMBL5545590 0.83 GSK3B (0.35) ADORA1GSK3BGSK3A
SCHEMBL5545504 0.83 GAA (0.43) ILKADORA1GSK3BGSK3A
SCHEMBL5543665 0.82 GAA (0.40) MEN1KMT2AGSK3BGSK3AALDH1A1
SCHEMBL3522887 0.81 SYK (0.34) ADORA1GSK3BGSK3A
SCHEMBL5543598 0.81 HSD17B10 (0.43) ADORA1GSK3BGSK3ACYP2D6HSD17B10
SCHEMBL3525674 0.81 GSK3B (0.42) ADORA1GSK3BGSK3AKDM4ETSHR
SCHEMBL5550117 0.81 GAA (0.39) MEN1KMT2AGSK3BGSK3AALDH1A1
SCHEMBL5545643 0.81 GSK3B (0.34) ADORA1GSK3BGSK3A
SCHEMBL5545560 0.80 GSK3A (0.37) GSK3BGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed