SCHEMBL5545504

SCHEMBL5545504

CC(C)(C)c1cn2c(=O)[nH]nc2c(NCCCC(=O)O)n1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.43
GSK3A P49840 15/20 0.36
GSK3B P49841 15/20 0.36
SYK P43405 1/20 0.36
ILK Q13418 1/20 0.35
CDC25A P30304 1/20 0.34
CDC25B P30305 1/20 0.34
ADORA1 P30542 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5550117 0.96 GAA (0.39) GAAGSK3AGSK3BSYKCDC25A
SCHEMBL3521844 0.83 MAT2A (0.38) GSK3AGSK3B
SCHEMBL5550132 0.83 ILK (0.35) GSK3AGSK3BILKADORA1
SCHEMBL5545643 0.80 GSK3B (0.34) GSK3AGSK3BADORA1
SCHEMBL5548899 0.78 GSK3B (0.32) GSK3AGSK3BADORA1
SCHEMBL5543493 0.76 GSK3B (0.50) GSK3AGSK3BADORA1
SCHEMBL5550070 0.74 GSK3A (0.50) GSK3AGSK3B
SCHEMBL3529299 0.73 GSK3B (0.41) GSK3AGSK3BADORA1
SCHEMBL5550039 0.72 GSK3A (0.46) GSK3AGSK3BADORA1
SCHEMBL3523483 0.72 NPC1 (0.41) ILKADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed