Delanzomib

Delanzomib

SCHEMBL555047

CC(C)C[C@H](NC(=O)[C@@H](NC(=O)c1cccc(-c2ccccc2)n1)[C@@H](C)O)B(O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 12/20 1.00
PSMB1 P20618 5/20 1.00
PSMB8 P28062 5/20 1.00
PSMB9 P28065 5/20 1.00
PSMB10 P40306 5/20 1.00
PSMB2 P49721 5/20 1.00
ELANE P08246 2/20 1.00
CTSG P08311 2/20 1.00
CMA1 P23946 2/20 1.00
CYP3A4 P08684 1/20 1.00
CNR2 P34972 4/20 0.62
CLPP Q16740 2/20 0.53
LONP1 P36776 5/20 0.49
PSMB11 A5LHX3 4/20 0.49
PSMA7 O14818 4/20 0.49
PSMA1 P25786 4/20 0.49
PSMA2 P25787 4/20 0.49
PSMA3 P25788 4/20 0.49
PSMA4 P25789 4/20 0.49
PSMA5 P28066 4/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Delanzomib SCHEMBL18331130 1.00 PSMB5 (1.00) PSMB5PSMB1PSMB8PSMB9PSMB10
Delanzomib SCHEMBL29409193 1.00 PSMB5 (1.00) PSMB5PSMB1PSMB8PSMB9PSMB10
Delanzomib SCHEMBL20408479 1.00 PSMB5 (1.00) PSMB5PSMB1PSMB8PSMB9PSMB10
Delanzomib SCHEMBL19813892 1.00 PSMB5 (1.00) PSMB5PSMB1PSMB8PSMB9PSMB10
Delanzomib SCHEMBL23651269 1.00 PSMB5 (1.00) PSMB5PSMB1PSMB8PSMB9PSMB10
Delanzomib SCHEMBL23693013 1.00 PSMB5 (1.00) PSMB5PSMB1PSMB8PSMB9PSMB10
Delanzomib SCHEMBL13386470 1.00 PSMB5 (1.00) PSMB5PSMB1PSMB8PSMB9PSMB10
Delanzomib SCHEMBL13386388 1.00 PSMB5 (1.00) PSMB5PSMB1PSMB8PSMB9PSMB10
Delanzomib SCHEMBL13386473 1.00 PSMB5 (1.00) PSMB5PSMB1PSMB8PSMB9PSMB10
Delanzomib SCHEMBL18388691 1.00 PSMB5 (1.00) PSMB5PSMB1PSMB8PSMB9PSMB10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1986 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260130990-A1 METHODS FOR IMPROVED THERAPEUTIC USE OF RECOMBINANT AAV ULTRAGENYX PHARMACEUTICAL INC (US) 2026-05-14 US claimed
US-20260130856-A1 LIPOSOME COMPOSITIONS FOR DELIVERY OF COMPOUNDS AND METHODS THEREOF NANOTECH PHARMA INC (US) 2026-05-14 US claimed
US-20260102375-A1 PHARMACEUTICAL COMBINATIONS FOR TREATING CANCER PURDUE PHARMACEUTICAL PRODUCTS L.P. (US) 2026-04-16 US claimed
US-20260069567-A1 Pharmaceutical Combinations For The Treatment Of Cancer PRESAGE BIOSCIENCES, INC. (US) 2026-03-12 US claimed
EP-4706663-A2 FAP-ACTIVATED PROTEASOME INHIBITORS FOR TREATING SOLID TUMORS Trustees Of Tufts College (US) 2026-03-11 EP claimed
EP-3897625-B1 COMPOUNDS FOR TREATING LYMPHOMA OR A T-CELL MALIGNANT DISEASE MUNDIPHARMA INTERNATIONAL CORPORATION LTD (BM) 2026-01-28 EP claimed
EP-4667458-A1 PHARMACEUTICAL COMPOSITION FOR TREATMENT OF CANCER, COMPRISING SOS1 INHIBITOR AND ANTICANCER DRUG Kanaph Therapeutics Inc. (KR) 2025-12-24 EP claimed
US-20250367304-A1 FAP-ACTIVATED PROTEASOME INHIBITORS FOR TREATING SOLID TUMORS TUFTS COLLEGE (US) 2025-12-04 US claimed
EP-3436002-B1 PHARMACEUTICAL COMBINATIONS FOR THE TREATMENT OF CANCER PRESAGE BIOSCIENCES INC (US) 2025-11-05 EP claimed
EP-3897626-B1 TINOSTAMUSTINE FOR TREATING MULTIPLE MYELOMA MUNDIPHARMA INTERNATIONAL CORPORATION LTD (BM) 2025-09-10 EP claimed
EP-3994132-A1 TYROSINE KINASE NON-RECEPTOR 1 (TNK1) INHIBITORS AND USES THEREOF Sumitomo Dainippon Pharma Oncology, Inc. (US) 2022-05-11 EP claimed
WO-2022094262-A1 FAP-ACTIVATED SERUM EXTENDED HALF-LIFE THERAPEUTIC CONJUGATES AVACTA LIFE SCIENCES LIMITED (GB) 2022-05-05 WO claimed
EP-3768265-B1 NEW CENTRALLY-ACTIVE GHRELIN AGONIST AND MEDICAL USES THEREOF HELSINN HEALTHCARE SA (CH) 2022-05-04 EP claimed
US-11320422-B2 Inhibition of protein degradation for improved production LONZA LTD. (CH) 2022-05-03 US claimed
CN-114302878-A Tyrosine kinase non-receptor 1(TNK1) inhibitors and uses thereof 大日本住友制药肿瘤公司 2022-04-08 CN claimed
WO-2022032132-A1 ADVANTAGEOUS THERAPIES FOR DISORDERS MEDIATED BY IKAROS OR AIOLOS C4 THERAPEUTICS, INC. (US) 2022-02-10 WO claimed
EP-1660507-B2 PROTEASOME INHIBITORS AND METHODS OF USING THE SAME MILLENNIUM PHARM INC (US) 2017-01-04 EP claimed
US-20150184246-A1 BIOMARKERS OF RESPONSE TO PROTEASOME INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2015-07-02 US claimed
EP-1660507-B9 PROTEASOME INHIBITORS AND METHODS OF USING THE SAME CEPHALON INC (US) 2010-03-24 EP claimed
EP-1660507-B1 PROTEASOME INHIBITORS AND METHODS OF USING THE SAME CEPHALON INC (US) 2009-08-05 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260102375-A1 PHARMACEUTICAL COMBINATIONS FOR TREATING CANCER PSMB5, PSMD5, PSMA5 PSMB5 1/4885PSMB1 16/4885PSMB8 32/4885
US-20150184246-A1 BIOMARKERS OF RESPONSE TO PROTEASOME INHIBITORS PSME3, PSMB1, PSMB4 PSMB5 19/4885PSMB1 2/4885PSMB8 21/4885
US-20260130856-A1 LIPOSOME COMPOSITIONS FOR DELIVERY OF COMPOUNDS AND METHODS THEREOF SGMS2, SGMS1, LIPA PSMB5 2603/4885PSMB1 1727/4885PSMB8 1379/4885
US-20250367304-A1 FAP-ACTIVATED PROTEASOME INHIBITORS FOR TREATING SOLID TUMORS FAP, PSMA1, PSMB1 PSMB5 16/4885PSMB1 3/4885PSMB8 18/4885
US-20260069567-A1 Pharmaceutical Combinations For The Treatment Of Cancer BCL6, BCL6B, BCL9 PSMB5 304/4885PSMB1 189/4885PSMB8 160/4885
US-20260130990-A1 METHODS FOR IMPROVED THERAPEUTIC USE OF RECOMBINANT AAV ICOS, ICOSLG, LY6K PSMB5 2120/4885PSMB1 882/4885PSMB8 677/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.