SCHEMBL5553553

SCHEMBL5553553

CCCc1nc(CC)sc1C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 1/20 0.34
AGTR2 P50052 1/20 0.34
ALDH1A1 P00352 3/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
NPC1 O15118 3/20 0.33
RAB9A P51151 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HSP90AA1 P07900 1/20 0.33
GAA P10253 1/20 0.32
MAPK1 P28482 1/20 0.32
GPR35 Q9HC97 5/20 0.31
GABRP O00591 2/20 0.31
GABRD O14764 2/20 0.31
GABRA1 P14867 2/20 0.31
GABRB1 P18505 2/20 0.31
GABRG2 P18507 2/20 0.31
GABRB3 P28472 2/20 0.31
GABRA5 P31644 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9643784 0.91 ALDH1A1 (0.36) AGTR1AGTR2ALDH1A1HPGDTSHR
SCHEMBL5557234 0.90 GABRP (0.42) ALDH1A1TSHRRAB9AMEN1KMT2A
SCHEMBL9642917 0.87 RAB9A (0.40) ALDH1A1HPGDTSHRNPC1RAB9A
SCHEMBL9642897 0.86 MEN1 (0.37) ALDH1A1HPGDTSHRNPC1RAB9A
Hydrochloric Acid SCHEMBL9528440 0.85 RAB9A (0.39) ALDH1A1HPGDTSHRNPC1RAB9A
SCHEMBL10441533 0.83 GABRP (0.42) ALDH1A1TSHRMEN1KMT2AGAA
SCHEMBL9644276 0.82 ALDH1A1 (0.38) ALDH1A1HPGDTSHRNPC1RAB9A
SCHEMBL9643713 0.82 ALDH1A1 (0.34) ALDH1A1HPGDTSHRNPC1RAB9A
SCHEMBL10268826 0.81 NPC1 (0.46) ALDH1A1HPGDNPC1RAB9AKDM4E
SCHEMBL9643993 0.81 GABRP (0.43) ALDH1A1TSHRMEN1KMT2AGPR35

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120108565-A1 PYRROLE CARBOXYLIC ACID DERIVATIVES AS ANTIBACTERIAL AGENTS RANBAXY LABORATORIES LIMITED (IN) 2012-05-03 US disclosed
US-5136042-A PROCESS FOR THE PREPARATION OF THIAZOLECARBOXYLIC ACID CHLORIDES MITSUI TOATSU CHEMICALS, INC. (JP) 1992-08-04 US disclosed
EP-0377750-A1 PROCESS FOR PREPARING THIAZOLECARBOXYLIC ACID CHLORIDES MITSUI CHEMICALS, INC. (JP) 1990-07-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120108565-A1 PYRROLE CARBOXYLIC ACID DERIVATIVES AS ANTIBACTERIAL AGENTS POLI, POLB, POLA1 AGTR1 1723/4885AGTR2 2270/4885ALDH1A1 2042/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.