SCHEMBL5553765

SCHEMBL5553765

COc1cc2c(OC(C)=O)c(C)n(C(=O)c3ccc(F)cc3)c2cc1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 4/20 0.45
AKR1C2 P52895 4/20 0.45
PTGS2 P35354 3/20 0.43
PTGS1 P23219 1/20 0.42
GAA P10253 1/20 0.40
PDE10A Q9Y233 1/20 0.39
MAPT P10636 2/20 0.37
TUBB4A P04350 1/20 0.37
TUBB P07437 1/20 0.37
TUBA3C P0DPH7 1/20 0.37
TUBA1B P68363 1/20 0.37
TUBA4A P68366 1/20 0.37
TUBB4B P68371 1/20 0.37
TUBB3 Q13509 1/20 0.37
TUBB2A Q13885 1/20 0.37
TUBB8 Q3ZCM7 1/20 0.37
TUBA3E Q6PEY2 1/20 0.37
TUBA1A Q71U36 1/20 0.37
TUBA1C Q9BQE3 1/20 0.37
TUBB6 Q9BUF5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5560537 0.89 AKR1C3 (0.47) AKR1C3AKR1C2PTGS2PTGS1KDM4E
SCHEMBL5822660 0.83 AKR1C3 (0.65) AKR1C3AKR1C2PTGS2PTGS1MAPT
SCHEMBL5798784 0.80 PTGS2 (0.66) AKR1C3AKR1C2PTGS2PTGS1MAPT
SCHEMBL5553811 0.80 MAPT (0.40) AKR1C3AKR1C2PTGS2GAAMAPT
SCHEMBL5800794 0.80 PTGS2 (0.37) AKR1C3AKR1C2PTGS2PTGS1ABCB1
SCHEMBL3002102 0.79 AKR1C3 (0.72) AKR1C3AKR1C2PTGS2PTGS1MAPT
SCHEMBL2002678 0.79 AKR1C3 (0.47) AKR1C3AKR1C2PTGS2PTGS1LMNA
SCHEMBL5800598 0.79 AKR1C3 (0.43) AKR1C3AKR1C2PTGS2GAAMAPT
SCHEMBL5823303 0.79 AKR1C3 (0.43) AKR1C3AKR1C2PTGS2PTGS1KDM4E
SCHEMBL15062379 0.78 PTGS1 (0.31) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
WO-2006050120-A2 SYNTHESIS OF COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2006-05-11 WO disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed