SCHEMBL5554335

SCHEMBL5554335

CCOC(=O)[C@@H](C)c1c(C)n(C(=O)c2ccc(F)c(F)c2)c2ccc(O)c(F)c12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
PTGS2 P35354 6/20 0.34
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NR1H4 Q96RI1 3/20 0.33
AKR1C3 P42330 2/20 0.33
AKR1C2 P52895 2/20 0.33
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32
CHRM1 P11229 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5554332 1.00 ALDH1A1 (0.35) ALDH1A1PTGS2CA12CA1CA2
SCHEMBL5800238 0.93 PTGS2 (0.37) ALDH1A1PTGS2MEN1KMT2AAKR1C3
SCHEMBL5800235 0.93 PTGS2 (0.37) ALDH1A1PTGS2MEN1KMT2AAKR1C3
SCHEMBL5808994 0.91 PTGS2 (0.35) PTGS2AKR1C3AKR1C2PSEN1PSEN2
SCHEMBL5808998 0.91 PTGS2 (0.35) PTGS2AKR1C3AKR1C2PSEN1PSEN2
SCHEMBL5824143 0.89 APP (0.38) PTGS2MEN1KMT2AAKR1C3AKR1C2
SCHEMBL5797670 0.89 PTGS2 (0.43) PTGS2AKR1C3AKR1C2
SCHEMBL5797673 0.89 PTGS2 (0.43) PTGS2AKR1C3AKR1C2
SCHEMBL5800263 0.88 TSHR (0.39) PTGS2AKR1C3AKR1C2PSEN1PSEN2
SCHEMBL5800266 0.88 TSHR (0.39) PTGS2AKR1C3AKR1C2PSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
WO-2006050120-A2 SYNTHESIS OF COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2006-05-11 WO disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed