SCHEMBL5554440

SCHEMBL5554440

CC[C@@H](C)c1cc2c(c(F)c1O)c(OC(C)=O)c(C)n2C(=O)c1ccc(F)c(F)c1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
AKR1C3 P42330 2/20 0.31
AKR1C2 P52895 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5560065 0.93 PTGS2 (0.31) PTGS2AKR1C3AKR1C2
SCHEMBL5813879 0.89 AKR1C3 (0.38) PTGS2MEN1KMT2AAKR1C3AKR1C2
SCHEMBL5554427 0.86 MEN1 (0.32) PTGS2MEN1KMT2A
SCHEMBL5560536 0.85 KMT2A (0.36) PTGS2MEN1KMT2AAKR1C3AKR1C2
SCHEMBL5554454 0.83 PTGS2 (0.40) PTGS2MEN1KMT2AAKR1C3AKR1C2
SCHEMBL5558659 0.80 PTGS2 (0.39) PTGS2AKR1C3AKR1C2
SCHEMBL5560071 0.80 PTGS2 (0.39) PTGS2AKR1C3AKR1C2
SCHEMBL5554202 0.77 TACR3 (0.33) PTGS2AKR1C3AKR1C2
SCHEMBL5558629 0.77 AKR1C3 (0.37) PTGS2AKR1C3AKR1C2
SCHEMBL5559390 0.77 AKR1C3 (0.42) PTGS2MEN1KMT2AAKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed