SCHEMBL5555467

SCHEMBL5555467

CCc1c(CO)nn(C(C)C)c1Oc1ccccc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPO P05164 3/20 0.36
HTT P42858 3/20 0.35
NPSR1 Q6W5P4 3/20 0.35
HRH3 Q9Y5N1 1/20 0.34
HTR2C P28335 3/20 0.33
HTR2A P28223 1/20 0.33
HTR2B P41595 1/20 0.33
KMT2A Q03164 1/20 0.33
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
RHEB Q15382 1/20 0.32
XIAP P98170 1/20 0.32
CXCL8 P10145 1/20 0.32
HTR1A P08908 1/20 0.32
POLB P06746 1/20 0.32
ALDH1A1 P00352 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5560668 0.80 MAPT (0.37) MPOHTTHRH3KMT2AXIAP
SCHEMBL5561831 0.80 NPBWR1 (0.35) HRH3HTR2ASLC6A2SLC6A4SLC6A3
SCHEMBL5560864 0.78 CYP1A2 (0.31) MPOPOLBCYP1A2CYP2C19MAPT
SCHEMBL5555674 0.71 EPAS1 (0.41) HRH3
SCHEMBL5560726 0.71 CYP1A2 (0.41) HRH3HTR2ASLC6A2SLC6A4SLC6A3
SCHEMBL14471432 0.69 RHEB (0.37) HTTNPSR1KMT2ASLC6A2SLC6A4
SCHEMBL5562173 0.69 EPAS1 (0.34) MPOPOLBCYP1A2CYP2C19
SCHEMBL5555486 0.68 CYP1A2 (0.33) POLBCYP1A2CYP2C19
SCHEMBL5561648 0.67 EPAS1 (0.32) POLBCYP1A2CYP2C19
SCHEMBL5560810 0.67 EPAS1 (0.36) POLBCYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1597235-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2007-08-15 EP disclosed
US-7241794-B2 Nonnucleoside reverse transcriptase inhibitors ROCHEPALO ALTO LLC (US) 2007-07-10 US disclosed
US-7241794-B2 Nonnucleoside reverse transcriptase inhibitors ROCHEPALO ALTO LLC (US) 2007-07-10 US disclosed