SCHEMBL5555674

SCHEMBL5555674

CCc1c(CO)nn(C(C)C)c1Oc1cccc(C#N)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 3/20 0.41
MGLL Q99685 2/20 0.39
HRH3 Q9Y5N1 1/20 0.39
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
NR1H4 Q96RI1 1/20 0.35
PIK3CD O00329 1/20 0.34
ABL1 P00519 1/20 0.34
EGFR P00533 1/20 0.34
HCK P08631 1/20 0.34
SRC P12931 1/20 0.34
KDR P35968 1/20 0.34
PIK3CA P42336 1/20 0.34
MTOR P42345 1/20 0.34
PIK3CG P48736 1/20 0.34
EPHB4 P54760 1/20 0.34
PRKDC P78527 1/20 0.34
PI4KB Q9UBF8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5561726 0.89 KCNH2 (0.40) EPAS1
SCHEMBL5560933 0.86 PGR (0.39) HRH3KDRSCN9A
SCHEMBL5555878 0.84 EPAS1 (0.38) EPAS1MGLLHRH3PDE4APDE4B
SCHEMBL5562337 0.84 KCNH2 (0.45) EPAS1
SCHEMBL5555927 0.83 CYP1A2 (0.40) MGLLHRH3
SCHEMBL5561831 0.77 NPBWR1 (0.35) MGLLHRH3MCHR1
SCHEMBL5560726 0.76 CYP1A2 (0.41) MGLLHRH3EGFR
SCHEMBL5562024 0.76 KCNH2 (0.43) EPAS1
SCHEMBL5560864 0.76 CYP1A2 (0.31) EPAS1
SCHEMBL5560668 0.76 MAPT (0.37) MGLLHRH3MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1597235-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2007-08-15 EP disclosed
US-7241794-B2 Nonnucleoside reverse transcriptase inhibitors ROCHEPALO ALTO LLC (US) 2007-07-10 US disclosed
US-7241794-B2 Nonnucleoside reverse transcriptase inhibitors ROCHEPALO ALTO LLC (US) 2007-07-10 US disclosed