SCHEMBL5560668

SCHEMBL5560668

CCc1c(CO)nn(C(C)C)c1Oc1ccc(Cl)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
NOTUM Q6P988 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
LTA4H P09960 2/20 0.35
CYP2D6 P10635 2/20 0.34
CYP2C9 P11712 2/20 0.34
MPO P05164 2/20 0.33
ENPP3 O14638 1/20 0.32
ALPL P05186 1/20 0.32
ENPP1 P22413 1/20 0.32
XIAP P98170 1/20 0.32
MGLL Q99685 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
NPBWR1 P48145 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5560864 0.87 CYP1A2 (0.31) MAPTMPOCYP1A2CYP2C19
SCHEMBL5561831 0.86 NPBWR1 (0.35) MGLLHRH3NPBWR1MCHR1
SCHEMBL5555927 0.85 CYP1A2 (0.40) SMN1; SMN2CYP2C9MGLLCYP1A2CYP2C19
SCHEMBL5560933 0.84 PGR (0.39) KDM4EHRH3
SCHEMBL5555467 0.80 MPO (0.36) MAPTHTTCYP2C9MPOXIAP
SCHEMBL5562173 0.79 EPAS1 (0.34) MPOCYP1A2CYP2C19
SCHEMBL5560726 0.78 CYP1A2 (0.41) SMN1; SMN2CYP2C9MGLLCYP1A2CYP2C19
SCHEMBL5560810 0.76 EPAS1 (0.36) CYP1A2CYP2C19
SCHEMBL5561648 0.76 EPAS1 (0.32) CYP1A2CYP2C19
SCHEMBL5555325 0.74 CYP1A2 (0.31) MPOCYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1597235-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2007-08-15 EP disclosed
US-7241794-B2 Nonnucleoside reverse transcriptase inhibitors ROCHEPALO ALTO LLC (US) 2007-07-10 US disclosed
US-7241794-B2 Nonnucleoside reverse transcriptase inhibitors ROCHEPALO ALTO LLC (US) 2007-07-10 US disclosed