SCHEMBL5555856

SCHEMBL5555856

CCOC(=O)Cc1nn(C(C)C)c(Oc2cc(Cl)cc(Cl)c2)c1CC

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.37
KDM4E B2RXH2 5/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.34
RECQL P46063 1/20 0.34
ALDH1A1 P00352 3/20 0.34
CCNE2 O96020 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
HPGD P15428 2/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
FPR1 P21462 1/20 0.32
KMT2A Q03164 1/20 0.32
HTT P42858 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PTGS2 P35354 1/20 0.32
MAPK1 P28482 2/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5561735 0.90 MAPT (0.37) MAPTL3MBTL1SMN1; SMN2RECQLALDH1A1
SCHEMBL14453992 0.89 MAPT (0.36) MAPTL3MBTL1CYP1A2POLBCYP2C19
SCHEMBL5557512 0.88 PTGDR2 (0.33) MAPTCYP1A2POLBCYP2C19PTGDR2
SCHEMBL5556006 0.88 PTGDR2 (0.41) MAPTCYP1A2POLBCYP2C19PTGDR2
SCHEMBL5556070 0.87 SIRT1 (0.34) MAPTALDH1A1CYP1A2POLBCYP2C19
SCHEMBL5562406 0.85 CARM1 (0.33) MAPTRECQLPTGS2PTGDR2
SCHEMBL14454008 0.83 CARM1 (0.33) MAPTPTGDR2
SCHEMBL5560864 0.83 CYP1A2 (0.31) MAPTCYP1A2POLBCYP2C19
SCHEMBL5561748 0.82 MAPT (0.42) MAPTKDM4EL3MBTL1ALDH1A1HPGD
SCHEMBL5561941 0.82 MAPT (0.32) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1597235-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2007-08-15 EP disclosed
US-7241794-B2 Nonnucleoside reverse transcriptase inhibitors ROCHEPALO ALTO LLC (US) 2007-07-10 US disclosed
US-7241794-B2 Nonnucleoside reverse transcriptase inhibitors ROCHEPALO ALTO LLC (US) 2007-07-10 US disclosed