SCHEMBL5558835

SCHEMBL5558835

COc1c(Cl)cc2c(c1C)c(OC(C)=O)c(C)n2C(=S)c1ccc(C)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.38
TAS1R3 Q7RTX0 3/20 0.34
TAS1R1 Q7RTX1 3/20 0.34
TAS1R2 Q8TE23 2/20 0.34
KMT2A Q03164 2/20 0.33
LMNA P02545 2/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
PTGS2 P35354 2/20 0.31
PTGS1 P23219 1/20 0.31
TP53 P04637 1/20 0.31
POLB P06746 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
TUBB4A P04350 1/20 0.31
TUBB P07437 1/20 0.31
TUBA3C P0DPH7 1/20 0.31
TUBA1B P68363 1/20 0.31
TUBA4A P68366 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5554313 0.86 ABCB11 (0.38) ABCB11PTGS2PTGS1AKR1C3AKR1C2
SCHEMBL5554035 0.85 ABCB11 (0.33) ABCB11TAS1R3TAS1R1TAS1R2KMT2A
SCHEMBL5560622 0.85 ABCB11 (0.33) ABCB11TAS1R3TAS1R1TAS1R2PTGS2
SCHEMBL5556641 0.85 ABCB11 (0.33) ABCB11TAS1R3TAS1R1TAS1R2KMT2A
SCHEMBL5558673 0.81 PTGS2 (0.43) ABCB11KMT2ALMNAMEN1PTGS2
SCHEMBL5559012 0.81
SCHEMBL5558850 0.76 AKR1C3 (0.40) ABCB11LMNAPTGS2PTGS1TP53
SCHEMBL5813595 0.74 PTGS2 (0.46) PTGS2PTGS1
SCHEMBL5558610 0.68 PTGS2 (0.43) ABCB11KMT2ALMNAMEN1PTGS2
SCHEMBL5554224 0.68 AKR1C3 (0.35) ABCB11KMT2ALMNAMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed