SCHEMBL5560926

SCHEMBL5560926

CCc1c(CO)nn(CC)c1Oc1cc(Cl)cc(C#N)c1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.47
CYP3A4 P08684 3/20 0.34
CNR1 P21554 4/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.32
EPAS1 Q99814 3/20 0.31
VEGFA P15692 1/20 0.31
ARNT P27540 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5560603 0.91 KCNH2 (0.45) KCNH2CYP3A4CNR1PTGDR2
SCHEMBL5561074 0.88 PTGDR2 (0.34) KCNH2PTGDR2MAPTKMT2A
SCHEMBL5562337 0.85 KCNH2 (0.45) KCNH2CYP3A4EPAS1VEGFAARNT
SCHEMBL5561581 0.83 PGR (0.41) MAPTKMT2A
SCHEMBL5555878 0.83 EPAS1 (0.38) EPAS1
SCHEMBL14454033 0.81 KCNH2 (0.43) KCNH2CYP3A4CNR1EPAS1VEGFA
SCHEMBL14454032 0.81 KCNH2 (0.41) KCNH2CYP3A4
SCHEMBL5561781 0.79 PTGDR2 (0.38) KCNH2PTGDR2MAPT
SCHEMBL5555445 0.79 CYP1A2 (0.41) KCNH2CYP3A4PTGDR2KMT2A
SCHEMBL5562279 0.79 GABRB3 (0.32) PTGDR2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1597235-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2007-08-15 EP disclosed
US-7241794-B2 Nonnucleoside reverse transcriptase inhibitors ROCHEPALO ALTO LLC (US) 2007-07-10 US disclosed