SCHEMBL5563990

SCHEMBL5563990

COC(=O)c1ccc(C(=O)NCCc2cccc(OC(F)(F)F)c2)s1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.53
HDAC3 O15379 1/20 0.53
HDAC4 P56524 1/20 0.53
HDAC1 Q13547 1/20 0.53
HDAC6 Q9UBN7 1/20 0.53
TRPV1 Q8NER1 2/20 0.53
KCNN4 O15554 1/20 0.47
NAMPT P43490 2/20 0.47
LMNA P02545 1/20 0.47
MAPK14 Q16539 1/20 0.46
RAB9A P51151 1/20 0.45
CLK1 P49759 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
CHRM2 P08172 1/20 0.44
CHRM1 P11229 1/20 0.44
CHRM3 P20309 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5565068 0.81 NPC1 (0.51) CNR1HDAC3HDAC4HDAC1HDAC6
SCHEMBL6455155 0.81 HDAC3 (0.65) HDAC3HDAC4HDAC1HDAC6NAMPT
SCHEMBL5560316 0.81 MRGPRX4 (0.49) HDAC3HDAC4HDAC1HDAC6TRPV1
SCHEMBL14100173 0.79 RAB9A (0.57) CNR1NAMPTLMNARAB9ACLK1
SCHEMBL3577619 0.79 TRPV1 (0.69) CNR1HDAC3HDAC4HDAC1HDAC6
SCHEMBL5565747 0.78 SMN1; SMN2 (0.50) HDAC3HDAC4HDAC1HDAC6NAMPT
SCHEMBL27422506 0.77 CNR1 (0.67) CNR1TRPV1NAMPTMAPK14CHRM2
SCHEMBL7643257 0.77 CNR1 (0.63) CNR1TRPV1NAMPTMAPK14CHRM2
SCHEMBL3391028 0.76 TRPV1 (0.65) CNR1TRPV1NAMPTMAPK14RAB9A
SCHEMBL6989302 0.75 CNR1 (0.58) CNR1HDAC3HDAC4HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1758880-A1 HYDROXAMATES, THEIR MANUFACTURE AND USE AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-07 EP disclosed
WO-2005121119-A1 HYDROXAMATES, THEIR MANUFACTURE AND USE AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO disclosed