SCHEMBL5564182

SCHEMBL5564182

O=c1c2ccccc2cc(N2CCNCC2)c2ccccc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 8/20 0.60
NCF1 P14598 5/20 0.57
HTR5A P47898 3/20 0.57
HTR3E A5X5Y0 2/20 0.57
HTR3B O95264 2/20 0.57
HTR3A P46098 2/20 0.57
HTR3D Q70Z44 2/20 0.57
HTR3C Q8WXA8 2/20 0.57
SIGMAR1 Q99720 2/20 0.57
CYP1A2 P05177 1/20 0.57
HTR1A P08908 1/20 0.57
CYP2D6 P10635 1/20 0.57
TSHR P16473 1/20 0.57
NFKB1 P19838 1/20 0.57
HTR1D P28221 1/20 0.57
HTR1B P28222 1/20 0.57
HTR2A P28223 1/20 0.57
HTR7 P34969 1/20 0.57
MTOR P42345 1/20 0.57
HSD17B10 Q99714 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9904943 0.84 PRKDC (0.53) HTR6NCF1KDM4EALDH1A1HPGD
SCHEMBL10994076 0.81 NCF1 (0.51) NCF1HTR3ALMNA
SCHEMBL5369146 0.78 HTR6 (0.68) HTR6NCF1HTR5AHTR3EHTR3B
SCHEMBL10566917 0.75 HTR6 (1.00) HTR6NCF1HTR5AHTR3EHTR3B
SCHEMBL3166780 0.73 HTR6 (1.00) HTR6NCF1HTR5AHTR3EHTR3B
SCHEMBL240244 0.73 HTR6 (1.00) HTR6NCF1HTR5AHTR3EHTR3B
SCHEMBL29385724 0.73 HTR6 (1.00) HTR6NCF1HTR5AHTR3EHTR3B
SCHEMBL6959807 0.72 HTR6 (0.72) HTR6NCF1HTR5AHTR3EHTR3B
SCHEMBL722215 0.72 BACE1 (0.55) HTR6NCF1HTR5AHTR3EHTR3B
SCHEMBL725003 0.72 HTR6 (0.49) HTR6NCF1HTR5AHTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1492794-B1 PIPERAZINE SUBSTITUTED ARYL BENZODIAZEPINES AND THEIR USE AS DOPAMINE RECEPTOR ANTAGONISTS FOR THE TREATMENT OF PSYCHOTIC DISORDERS LILLY CO ELI (US) 2007-12-12 EP disclosed