SCHEMBL5564338

SCHEMBL5564338

Cc1cc(NC(=O)C2(N)CC3CCC2O3)ccc1N1CCCCN1C

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.33
NPC1 O15118 1/20 0.33
HRH3 Q9Y5N1 5/20 0.33
MAPT P10636 2/20 0.32
GAA P10253 2/20 0.32
TP53 P04637 2/20 0.32
ALDH1A1 P00352 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
POLB P06746 1/20 0.32
F13A1 P00488 1/20 0.32
TGM2 P21980 1/20 0.32
EPHX2 P34913 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5565253 0.81 NPC1 (0.34) RAB9ANPC1HRH3MAPTGAA
SCHEMBL6454562 0.78 F10 (0.40) RAB9ANPC1ALDH1A1SMN1; SMN2MEN1
SCHEMBL5563297 0.75 GAA (0.37) RAB9ANPC1MAPTGAAALDH1A1
SCHEMBL5568419 0.71 NPY2R (0.42) RAB9ANPC1MAPTSMN1; SMN2
SCHEMBL5564703 0.69 ALDH1A1 (0.34) RAB9ANPC1HRH3MAPTGAA
SCHEMBL6454489 0.65 CTSL (0.39) RAB9ANPC1MAPTGAATP53
SCHEMBL6454350 0.65 F10 (0.39) RAB9ANPC1ALDH1A1SMN1; SMN2MEN1
SCHEMBL6454183 0.63 F10 (0.45) RAB9ANPC1MAPTALDH1A1SMN1; SMN2
SCHEMBL5504268 0.62 F10 (0.48)
SCHEMBL5563698 0.61 HRH3 (0.40) RAB9ANPC1HRH3MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1748997-A1 SUBSTITUTED THIOPHENE-2-CARBOXYLIC ACID AMIDES, THE PRODUCTION THEREOF AND THE USE THEREOF AS DRUGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-02-07 EP disclosed
WO-2005111013-A1 SUBSTITUTED THIOPHENE-2-CARBOXYLIC ACID AMIDES, THE PRODUCTION THEREOF AND THE USE THEREOF AS DRUGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-11-24 WO disclosed