SCHEMBL5564599

SCHEMBL5564599

[CH2]CCCCN1CCS(=O)(=O)CC1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.36
KMT2A Q03164 3/20 0.35
MEN1 O00255 1/20 0.35
HPGD P15428 1/20 0.34
PAOX Q6QHF9 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CNR2 P34972 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2016182 0.93 KMT2A (0.36) HRH3KMT2AMEN1HPGDPAOX
SCHEMBL356238 0.84 KMT2A (0.38) KMT2AMEN1HPGDCYP1A2CYP2C19
SCHEMBL2850740 0.78 PAOX (0.37) HRH3KMT2AMEN1HPGDPAOX
SCHEMBL11269259 0.78 KEAP1 (0.43) HRH3KMT2AMEN1
SCHEMBL12550619 0.78 GNAO1 (0.48) KMT2AMEN1CNR2
SCHEMBL1097457 0.77 KMT2A (0.37) HRH3KMT2AMEN1HPGDPAOX
SCHEMBL12550641 0.77 GNAO1 (0.52)
SCHEMBL12550633 0.77 PAOX (0.40) HRH3KMT2AMEN1HPGDPAOX
SCHEMBL12550618 0.77 GNAO1 (0.52)
SCHEMBL12550634 0.77 PAOX (0.40) HRH3KMT2AMEN1HPGDPAOX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1751165-A1 4-SUBSTITUTED 1,5-DIHYDRO-PYRIDO(3,2-B)INDOL-2-ONES Tibotec Pharmaceuticals Ltd. (IE) 2007-02-14 EP disclosed
WO-2005111044-A1 4-SUBSTITUTED-1,5-DIHYDRO-PYRIDO[3,2-B]INDOL-2-ONES TIBOTEC PHARMACEUTICALS LTD. (IE) 2005-11-24 WO disclosed