SCHEMBL5565147

SCHEMBL5565147

CC/C=C/C1=CC(C)(C)COc2cc(-c3ccc(F)cc3)ccc21

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.35
HTR2B P41595 1/20 0.35
TMEM97 Q5BJF2 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
NR3C1 P04150 1/20 0.30
PGR P06401 1/20 0.30
NR3C2 P08235 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2316040 0.82 ESR1 (0.42) PGR
SCHEMBL2316048 0.82 ESR1 (0.42) PGR
SCHEMBL3604572 0.78 RXRA (0.38)
SCHEMBL3601994 0.77 HDAC1 (0.35)
SCHEMBL3601992 0.77 HDAC1 (0.35)
SCHEMBL5559796 0.76 NOTUM (0.31)
SCHEMBL5563963 0.73 KCNH2 (0.32)
SCHEMBL2316043 0.70 HDAC1 (0.34) PGR
SCHEMBL5564928 0.70 CHRM5 (0.33) HTR1AHTR2BSIGMAR1
SCHEMBL1399921 0.64 FABP6 (0.38) PGRNR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1758876-A1 NEW 5-ALKENONE-3,3-DIMETHYL-BENZOXEPINES DERIVATIVES USEFUL FOR THE PREPARATION OF ANTIDIABETIC PENTADIENOIC ACIDS MERCK PATENT GmbH (DE) 2007-03-07 EP disclosed
WO-2006002721-A1 NEW 5-ALKENONE-3,3-DIMETHYL-BENZOXEPINES DERIVATIVES USEFUL FOR THE PREPARATION OF ANTIDIABETIC PENTADIENOIC ACIDS MERCK PATENT GMBH (DE) 2006-01-12 WO disclosed