SCHEMBL2316043

SCHEMBL2316043

CC(=O)CCC1=CC(C)(C)COc2cc(-c3ccc(F)cc3)ccc21

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 12/20 0.34
HDAC2 Q92769 12/20 0.34
HDAC3 O15379 10/20 0.34
PGR P06401 1/20 0.33
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
KDM4C Q9H3R0 2/20 0.32
LTB4R Q15722 1/20 0.32
LTB4R2 Q9NPC1 1/20 0.32
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2322133 0.84 ALDH1A1 (0.39) PGR
SCHEMBL2314405 0.81 HTR2B (0.39) HDAC1HDAC2HDAC3PGR
SCHEMBL2317591 0.80 CYP3A4 (0.43) PGRESR1ESR2
SCHEMBL2321527 0.77 IMPDH2 (0.31)
SCHEMBL2316316 0.77 AKR1B1 (0.36)
SCHEMBL2316048 0.76 ESR1 (0.42) HDAC1HDAC2HDAC3PGRESR1
SCHEMBL2316040 0.76 ESR1 (0.42) HDAC1HDAC2HDAC3PGRESR1
SCHEMBL2316362 0.75 HTR1A (0.34) PGR
SCHEMBL2314396 0.74 MAPT (0.34) PGR
SCHEMBL2319041 0.74 CYP3A4 (0.35) PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1609786-B1 5-alkenone-3,3-dimethyl-benzoxepines derivatives useful for the preparation of antidiabetic pentadienoic acids MERCK SANTE SAS (FR) 2011-08-03 EP claimed