SCHEMBL5567645

SCHEMBL5567645

COC=Cc1ccc2cc(-c3cc(-c4ccncc4)nnc3OC)n(C(=O)O)c2c1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SQOR Q9Y6N5 1/20 0.32
CYP1A1 P04798 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP1B1 Q16678 1/20 0.31
CYP3A4 P08684 1/20 0.31
APP P05067 1/20 0.30
MAPT P10636 1/20 0.30
CASP1 P29466 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5567642 1.00 SQOR (0.32) SQORCYP1A1CYP1A2CYP2D6CYP1B1
SCHEMBL5562545 0.90 MAPT (0.36) SQORAPPMAPTCASP1
SCHEMBL1750961 0.89 NR1H2 (0.40)
SCHEMBL1750963 0.89 NR1H2 (0.40)
SCHEMBL5561371 0.82 ROCK1 (0.33) SQORCYP3A4MAPTCASP1
SCHEMBL5562265 0.82 SQOR (0.36) SQORCYP3A4MAPTCASP1
SCHEMBL1750386 0.78 NR1H2 (0.40) MAPT
SCHEMBL5567692 0.77 PARP1 (0.36)
SCHEMBL5567828 0.77 KDM4E (0.40) CYP2D6CYP3A4
SCHEMBL5562320 0.76 CYP1A2 (0.37) CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1751141-A1 NOVEL PYRIDAZINONE DERIVATIVES AS INHIBITORS OF CDK2 Aventis Pharma S.A. (FR) 2007-02-14 EP disclosed
WO-2005111019-A1 NOVEL PYRIDAZINONE DERIVATIVES AS INHIBITORS OF CDK2 AVENTIS PHARMA S.A. (FR) 2005-11-24 WO disclosed