SCHEMBL5567692

SCHEMBL5567692

COc1nnc(-c2ccncc2)cc1-c1cc2ccc(CN3CCCCC3)cc2n1C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
LSS P48449 1/20 0.36
MCHR1 Q99705 1/20 0.36
POLB P06746 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
CYP46A1 Q9Y6A2 1/20 0.35
CHEK1 O14757 1/20 0.35
ACHE P22303 1/20 0.35
ACP1 P24666 2/20 0.34
ALK Q9UM73 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5562320 0.92 CYP1A2 (0.37) POLBHRH3ACHE
SCHEMBL1751633 0.89 NR1H2 (0.38) PARP1LSSMCHR1
SCHEMBL5562265 0.86 SQOR (0.36) MEN1KMT2ACYP46A1
SCHEMBL5561371 0.85 ROCK1 (0.33) MEN1KMT2ACYP46A1
SCHEMBL3427396 0.82 NR1H2 (0.38) PARP1LSSALK
SCHEMBL1750986 0.81 NR1H2 (0.38)
SCHEMBL5562322 0.81 MKNK1 (0.32)
SCHEMBL5562545 0.79 MAPT (0.36)
SCHEMBL5567642 0.77 SQOR (0.32)
SCHEMBL5567645 0.77 SQOR (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1751141-A1 NOVEL PYRIDAZINONE DERIVATIVES AS INHIBITORS OF CDK2 Aventis Pharma S.A. (FR) 2007-02-14 EP disclosed
WO-2005111019-A1 NOVEL PYRIDAZINONE DERIVATIVES AS INHIBITORS OF CDK2 AVENTIS PHARMA S.A. (FR) 2005-11-24 WO disclosed