SCHEMBL5568564

SCHEMBL5568564

C=CCOC(=O)Nc1c(NCC2CCC3(CCC3)CC2)nc(C#N)nc1OCCC1CCN(C(=O)O)CC1

nearest known ligand 0.58

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSL P07711 20/20 0.58
CTSS P25774 16/20 0.58
KCNH2 Q12809 8/20 0.58
CTSK P43235 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3585874 0.91 CTSL (0.57) CTSLCTSSKCNH2CTSK
SCHEMBL5567274 0.82 CTSL (0.85) CTSLCTSSKCNH2CTSK
SCHEMBL3599719 0.81 CTSL (0.62) CTSLCTSSKCNH2CTSK
SCHEMBL5571480 0.79 CTSL (0.58) CTSLCTSSKCNH2CTSK
SCHEMBL5571484 0.78 CTSL (0.56) CTSLCTSSKCNH2CTSK
SCHEMBL3603514 0.76 CTSL (0.68) CTSLCTSSKCNH2CTSK
SCHEMBL5572278 0.74 CTSL (0.72) CTSLCTSSKCNH2CTSK
SCHEMBL3604323 0.74 CTSL (1.00) CTSLCTSSKCNH2CTSK
SCHEMBL3591605 0.73 CTSL (0.81) CTSLCTSSKCNH2CTSK
SCHEMBL3605017 0.73 GPR119 (0.39) CTSLCTSSKCNH2CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781623-A1 COMPOUNDS AND COMPOSITIONS USEFUL AS CATHEPSIN S INHIBITORS Novartis AG (CH) 2007-05-09 EP disclosed
WO-2006018284-A1 COMPOUNDS AND COMPOSITIONS USEFUL AS CATHEPSIN S INHIBITORS NOVARTIS AG (CH) 2006-02-23 WO disclosed