SCHEMBL5572278

SCHEMBL5572278

N#Cc1nc(NCC2CCC3(CCC3)CC2)cc(OCCC2CCN(C(=O)O)CC2)n1

nearest known ligand 0.72

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSL P07711 20/20 0.72
CTSS P25774 16/20 0.72
CTSK P43235 4/20 0.72
KCNH2 Q12809 7/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3585558 0.90 CTSL (0.70) CTSLCTSSCTSKKCNH2
SCHEMBL3599733 0.88 CTSL (0.93) CTSLCTSSCTSKKCNH2
SCHEMBL5567274 0.78 CTSL (0.85) CTSLCTSSCTSKKCNH2
SCHEMBL5571090 0.78 CTSS (0.46) CTSLCTSSCTSK
SCHEMBL5571484 0.75 CTSL (0.56) CTSLCTSSCTSKKCNH2
SCHEMBL5571480 0.75 CTSL (0.58) CTSLCTSSCTSKKCNH2
SCHEMBL5568564 0.74 CTSL (0.58) CTSLCTSSCTSKKCNH2
SCHEMBL3603514 0.72 CTSL (0.68) CTSLCTSSCTSKKCNH2
SCHEMBL3601032 0.71 CTSL (0.63) CTSLCTSSCTSKKCNH2
SCHEMBL3604323 0.69 CTSL (1.00) CTSLCTSSCTSKKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781623-A1 COMPOUNDS AND COMPOSITIONS USEFUL AS CATHEPSIN S INHIBITORS Novartis AG (CH) 2007-05-09 EP disclosed
WO-2006018284-A1 COMPOUNDS AND COMPOSITIONS USEFUL AS CATHEPSIN S INHIBITORS NOVARTIS AG (CH) 2006-02-23 WO disclosed