SCHEMBL5571013

SCHEMBL5571013

c1ccc2c(-c3c[nH]c4ccccc34)cncc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.53
IMPDH2 P12268 1/20 0.53
MAPK1 P28482 1/20 0.53
TDO2 P48775 4/20 0.52
ALDH1A1 P00352 2/20 0.51
MAPT P10636 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
LMNA P02545 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
GPR55 Q9Y2T6 1/20 0.51
PDGFRB P09619 2/20 0.51
PDGFRA P16234 1/20 0.51
PRKCZ Q05513 2/20 0.47
KDR P35968 1/20 0.47
IKBKE Q14164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20873066 0.81 PRKCZ (0.64) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL1202543 0.79 IMPDH2 (0.63) HSD17B10IMPDH2MAPK1ALDH1A1MAPT
SCHEMBL25034156 0.79 MAPT (0.57) HSD17B10IMPDH2MAPK1TDO2ALDH1A1
SCHEMBL3291196 0.78 ALDH1A1 (0.53) HSD17B10IMPDH2MAPK1TDO2ALDH1A1
SCHEMBL15333384 0.78 MAOB (0.59) HSD17B10IMPDH2MAPK1TDO2ALDH1A1
SCHEMBL17738793 0.78 IKBKE (0.76) IKBKETBK1CDK5CDK5R1GSK3B
SCHEMBL1919056 0.77 IMPDH2 (0.58) HSD17B10IMPDH2MAPK1TDO2ALDH1A1
SCHEMBL25034154 0.75 KDR (0.73) HSD17B10IMPDH2MAPK1TDO2PDGFRB
SCHEMBL10098237 0.73 PRKCZ (0.42) ALDH1A1MAPTSMN1; SMN2CYP3A4PRKCZ
SCHEMBL10806364 0.71 PRKCZ (0.69) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778639-A2 ARYL-AND HETEROARYL-SUBSTITUTED TETRAHYDROISOQUINOLINES AND USE THEREOF TO BLOCK REUPTAKE OF NOREPINEPHRINE, DOPAMINE, AND SEROTONIN AMR Technology, Inc. (US) 2007-05-02 EP disclosed
WO-2006020049-A2 ARYL-AND HETEROARYL-SUBSTITUTED TETRAHYDROISOQUINOLINES AND USE THEREOF TO BLOCK REUPTAKE OF NOREPINEPHRINE, DOPAMINE, AND SEROTONIN AMR TECHNOLOGY, INC. (US) 2006-02-23 WO disclosed