SCHEMBL5572920

SCHEMBL5572920

O=C(c1cccnc1)c1ncc(Cl)cc1[AsH2]

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.47
MAP2K1 Q02750 1/20 0.44
ALDH1A1 P00352 3/20 0.44
APP P05067 1/20 0.44
GAA P10253 1/20 0.44
HCAR3 P49019 1/20 0.44
HCAR2 Q8TDS4 1/20 0.44
PKM P14618 2/20 0.43
F7 P08709 1/20 0.42
F3 P13726 1/20 0.42
SARM1 Q6SZW1 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.42
SIRT6 Q8N6T7 1/20 0.42
SIRT1 Q96EB6 1/20 0.42
SIRT3 Q9NTG7 1/20 0.42
SIRT5 Q9NXA8 1/20 0.42
SIRT4 Q9Y6E7 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
KCNMA1 Q12791 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL306266 0.86 SMN1; SMN2 (0.47) SMN1; SMN2MAP2K1ALDH1A1APPGAA
SCHEMBL15268207 0.80 KCNMA1 (0.48) SMN1; SMN2MAP2K1ALDH1A1GAAMEN1
SCHEMBL305749 0.79 MAPT (0.51) SMN1; SMN2ALDH1A1MEN1KMT2AMAPT
SCHEMBL3409177 0.74 ALDH1A1 (0.50) SMN1; SMN2MAP2K1ALDH1A1APPGAA
SCHEMBL15646031 0.72 PKM (0.64) SMN1; SMN2ALDH1A1APPGAAHCAR3
SCHEMBL1242243 0.72 ALDH1A1 (0.71) MAP2K1ALDH1A1APPGAAHCAR3
SCHEMBL29915528 0.72 ALDH1A1 (0.71) MAP2K1ALDH1A1APPGAAHCAR3
SCHEMBL6665398 0.72 ALDH1A1 (0.59) SMN1; SMN2ALDH1A1APPGAAHCAR3
Hydrochloric Acid SCHEMBL27841975 0.70 ALDH1A1 (0.68) MAP2K1ALDH1A1APPGAAHCAR3
SCHEMBL18228667 0.70 ALDH1A1 (0.49) SMN1; SMN2MAP2K1ALDH1A1APPGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1838674-A2 HETEROARYL SULFONAMIDES AND CCR2 ChemoCentryx Inc (US) 2007-10-03 EP disclosed
WO-2006076644-A2 HETEROARYL SULFONAMIDES AND CCR2 CHEMOCENTRYX, INC. (US) 2006-07-20 WO disclosed