SCHEMBL5577182

SCHEMBL5577182

Cc1cc(O)c(Cl)cc1N1CCN(C(C)(C)C)CC1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 6/20 0.36
HSP90AB1 P08238 4/20 0.36
ALDH1A1 P00352 4/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
NPSR1 Q6W5P4 3/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ADAM17 P78536 1/20 0.34
ADAMTS5 Q9UNA0 1/20 0.34
USP2 O75604 2/20 0.33
MAPT P10636 2/20 0.33
TSHR P16473 2/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
AKR1C3 P42330 1/20 0.33
THRB P10828 1/20 0.32
HPGD P15428 1/20 0.31
HSD17B10 Q99714 1/20 0.31
MCOLN3 Q8TDD5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4930499 0.78 HSP90AA1 (0.51) HSP90AA1HSP90AB1ALDH1A1
SCHEMBL4931103 0.77 MEN1 (0.50) ALDH1A1MEN1KMT2ANPSR1SMN1; SMN2
SCHEMBL5577214 0.75 ALDH1A1 (0.34) ALDH1A1MEN1KMT2ANPSR1SMN1; SMN2
SCHEMBL12752842 0.69 ADRB1 (0.53) ALDH1A1LMNAHTTAKR1C3
SCHEMBL24309509 0.68 HSP90AA1 (0.54) HSP90AA1HSP90AB1MAPTTSHRHPGD
SCHEMBL1491177 0.68 GAA (0.54) ALDH1A1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL16432438 0.68 IGF1R (0.43) ALDH1A1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL11299409 0.68 MAPT (0.65) ALDH1A1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL24421699 0.68 ESR1 (0.43) ALDH1A1MEN1KMT2ANPSR1SMN1; SMN2
SCHEMBL11296569 0.68 MAPT (0.66) ALDH1A1MEN1KMT2ANPSR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1750727-A2 KINASE MODULATORS AND METHODS OF USE Exelixis, Inc. (US) 2007-02-14 EP disclosed
WO-2005117909-A2 KINASE MODULATORS AND METHODS OF USE EXELIXIS, INC. (US) 2005-12-15 WO disclosed